Perkin 1 Abstracts: Natural Product Synthesis Andrew Gunn Jacqueline E. Milne and Marcel de Puit pg 1-xii; DOI: 10.1039/b110868a |
Stoichiometric asymmetric processes Simon Jones pg 1; DOI: 10.1039/b009236n |
A chemoenzymatic synthesis of the 12-membered macrolide (–)-cladospolide A Martin G. Banwell Katrina A. Jolliffe David T. J. Loong Kenneth J. McRae and Filisaty Vounatsos pg 22; DOI: 10.1039/b110018a |
Inverse Wittig reaction of oxaphosphetenes formed by the [2+2] cycloaddition of arylphosphine oxides and dimethyl acetylenedicarboxylate (DMAD) György Keglevich Henrietta Forintos Tamás Körtvélyesi and László Tke pg 26; DOI: 10.1039/b108675h |
Phenyl group acceleration of [1,4] carbon-to-oxygen silicon-mediated elimination–rearrangement in -silyl sulfones. Synthesis of O-silylated cinnamyl alcohols Stefano Menichetti and Charles J. M. Stirling pg 28; DOI: 10.1039/b109805e |
Aryl H-phosphonates. Part 13. A new, general entry to aryl nucleoside phosphate and aryl nucleoside phosphorothioate diesters Jacek Cielak Jadwiga Jankowska Micha Sobkowski Magorzata Wenska Jacek Stawiski and Adam Kraszewski pg 31; DOI: 10.1039/b109373h |
On the optical activity of the 3-aryl-4-hydroxycoumarin isolated from Millettia griffoniana: molecular modelling and total synthesis Sébastien Combes Jean-Pierre Finet and Didier Siri pg 38; DOI: 10.1039/b108707j |
Influence of preparation procedure on polymer composition: synthesis and characterisation of polymethacrylates bearing -D-glucopyranoside and -D-galactopyranoside residues Moira Ambrosi Andrei S. Batsanov Neil R. Cameron Benjamin G. Davis Judith A. K. Howard and Rob Hunter pg 45; DOI: 10.1039/b108421f |
Photochemical transformations of 5-halogeno-4-thiouridines Grayna Wenska Katarzyna Taras-Goliska Katarzyna Lamparska-Kupsik Bohdan Skalski Maria Gdaniec and Zofia Gdaniec pg 53; DOI: 10.1039/b108380e |
Cascade radical synthesis of heteroarenes via iminyl radicals W. Russell Bowman Colin F. Bridge Philip Brookes Martin O. Cloonan and David C. Leach pg 58; DOI: 10.1039/b108323f |
4-Phenyloxazolidin-2-ones and isoindolin-1-ones: chiral auxiliaries for Diels–Alder reactions of N-substituted 1,3-dienes Helena McAlonan James P. Murphy Mark Nieuwenhuyzen Karen Reynolds Pakala K. S. Sarma Paul J. Stevenson and Norris Thompson pg 69; DOI: 10.1039/b108059h |
Diastereocontrolled synthesis of hydroxylated lactams Mark. D. Andrews Andrew G. Brewster and Mark G. Moloney pg 80; DOI: 10.1039/b108056n |
Synthesis of soluble halogenated aryloxy substituted indium phthalocyanines M. John Plater Adam Jeremiah and Grant Bourhill pg 91; DOI: 10.1039/b107689m |
Reductive cleavage of N-substituted aromatic amides as tert-butyl acylcarbamates Ulf Ragnarsson Leif Grehn Hernani L. S. Maia and Luis S. Monteiro pg 97; DOI: 10.1039/b107330n |
The effect of oxygen on the regioselectivity in the rhodium catalysed hydrosilylation of 1,3-dienes Magnus Gustafsson and Torbjörn Frejd pg 102; DOI: 10.1039/b106143g |
Controlled stepwise conversion of 2,4,6,8-tetrachloropyrimido[5,4-d]pyrimidine into 2,4,6,8-tetrasubstituted pyrimido[5,4-d]pyrimidines Julian S. Northen F. Thomas Boyle William Clegg Nicola J. Curtin Andrew J. Edwards Roger J. Griffin and Bernard T. Golding pg 108; DOI: 10.1039/b102224p |
The asymmetric Bischler–Napieralski reaction: preparation of 1,3,4-trisubstituted 1,2,3,4-tetrahydroisoquinolines Marcello Nicoletti David O'Hagan and Alexandra M. Z. Slawin pg 116; DOI: 10.1039/b106942j |
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis Gideon Grogan Alexis Carstairs Ian Jackson Denise McIntyre Alan Watt Sabine Flitsch and Nicholas Turner pg 2-vii; DOI: 10.1039/b111338k |
Photolabile protecting groups and linkers Christian G. Bochet pg 125; DOI: 10.1039/b009522m |
Synthesis of nornicotine, nicotine and other functionalised derivatives using solid-supported reagents and scavengers Ian R. Baxendale Gloria Brusotti Masato Matsuoka and Steven V. Ley pg 143; DOI: 10.1039/b109482n |
Use of a modified ring-switching strategy to synthesise the glutamate antagonist (2S)-2-amino-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)propionate and related compounds with two chiral centres Andrew Dinsmore Paul M. Doyle and Douglas W. Young pg 155; DOI: 10.1039/b109820a |
Metal triflates catalyzed efficient synthesis of 3,4-dihydro-2H-1-benzopyrans Jhillu S. Yadav Basi V. Subba Reddy M. Aruna Chenna Venugopal T. Ramalingam S. Kiran Kumar and Ajit C. Kunwar pg 165; DOI: 10.1039/b109538m |
-Methylene tetrazole-based peptidomimetics: synthesis and inhibition of HIV protease Barnaby C. H. May and Andrew D. Abell pg 172; DOI: 10.1039/b109128j |
Stereochemical considerations on the stereoselective cyclopropanation reactions of 3-aryl-2-phosphonoacrylates induced by the (–)-8-phenylmenthyl group as a chiral auxiliary Ryukichi Takagi Miki Hashizume Minoru Nakamura Shahnaz Begum Yoshikazu Hiraga Satoshi Kojima and Katsuo Ohkata pg 179; DOI: 10.1039/b108925k |
Two novel racemic synthetic approaches to LTB4 and LTB3 methyl esters Christine Gauthier Dominique Castet Yvan Ramondenc and Gérard Plé pg 191; DOI: 10.1039/b108847e |
Design and synthesis of N-nonpolar nucleobase dipeptides: application of the Ugi reaction for the preparation of dipeptides having fluoroarylalkyl groups appended to the nitrogen atom Biplab Kumar Das Norio Shibata and Yoshio Takeuchi pg 197; DOI: 10.1039/b108760f |
Regioselective synthesis of pyrazoles via the ring cleavage of 3-substituted N-alkylated 3-hydroxyisoindolin-1-ones Kyu-Tae Chang Yong Hyun Choi Seung-Ho Kim Yong-Jin Yoon and Woo Song Lee pg 207; DOI: 10.1039/b108485m |
Synthesis and alkylation reaction of 1-arylmethyleneamino- and 1-arylsulfonyl-5-hydroxy-1H-1,2,3-triazoles Yury A. Rozin Elena A. Savel'eva Yury Yu. Morzherin Wim Dehaen Suzanne Toppet Luc Van Meervelt and Vasily A. Bakulev pg 211; DOI: 10.1039/b108202g |
Synthesis of 6-alkyl analogues of the 1-azabicyclo[4.3.0]nonan-2-one system by a strategy of geminal acylation and Beckmann rearrangement Christine E. Elliott David O. Miller and D. Jean Burnell pg 217; DOI: 10.1039/b108164k |
Cleavage of cyclopropyl ketones mediated by alkylmercury(II) hydrides Pablo H. Di Chenna Andrés Ferrara Alberto A. Ghini and Gerardo Burton pg 227; DOI: 10.1039/b107258g |
Probing the mechanism of loss of carbon-20 in gibberellin biosynthesis. Synthesis of gibberellin 3,20-hemiacetal and 19,20-lactol analogues and their metabolism by a recombinant GA 20-oxidase Jane L. Ward Paul Gaskin Robert G. S. Brown Graham S. Jackson Peter Hedden Andy L. Phillips Christine L. Willis and Michael H. Beale pg 232; DOI: 10.1039/b106990j |
Parasite glycoconjugates. Part 12. Synthesis of deoxy, fluorodeoxy and aminodeoxy disaccharide phosphates, substrate analogues for the elongating -D-mannopyranosylphosphate transferase in the Leishmania Dmitry V. Yashunsky Yury E. Tsvetkov Michael A. J. Ferguson and Andrei V. Nikolaev pg 242; DOI: 10.1039/b106182h |
Kinetic resolution of amines with enantiopure 3-N,N-diacylaminoquinazolin-4(3H)-ones Abdullah G. Al-Sehemi Robert S. Atkinson and John Fawcett pg 257; DOI: 10.1039/b105917n |
Perkin 1 Abstracts: Natural Product Synthesis Andrew Gunn Jacqueline E. Milne Marcel de Puit and Duncan McArthur pg 3-ix; DOI: 10.1039/b200355b |
-Oxy sulfones and sulfoximines: versatile intermediates Fabrice Chemla pg 275; DOI: 10.1039/b009523k |
Synthesis of the first amine–cyanocarboxyboranes, isoelectronic analogues of -cyanocarboxylic acids Béla Györi Zoltán Berente Róbert Király and István Lázár pg 300; DOI: 10.1039/b111682g |
Facile synthesis of disubstituted and spiro five-membered benzosultams mediated by TMSCl–NaI–MeCN reagent Zhaopeng Liu Norio Shibata and Yoshio Takeuchi pg 302; DOI: 10.1039/b109832b |
Preparation of 1-phenylcyclohexa-2,5-diene-1-carboxylates and their use in free-radical mediated syntheses Paul A. Baguley Leon V. Jackson and John C. Walton pg 304; DOI: 10.1039/b110527m |
Synthesis of novel cyclophanes containing both benzo[1,2-b:5,4-b]difuran and naphthalene rings Kwanghee Koh Park Hongsan Lim Sun-Hyuk Kim and Dae Hyun Bae pg 310; DOI: 10.1039/b110312a |
Reaction of Herz salts with malononitrile: a general route to (6H-1,2,3-benzodithiazol-6-ylidene)malononitriles Panayiotis A. Koutentis and Charles W. Rees pg 315; DOI: 10.1039/b110024f |
Making conjugated connections to porphyrins: a comparison of alkyne, alkene, imine and azo links Thomas E. O. Screen Iain M. Blake Leigh H. Rees William Clegg Simon J. Borwick and Harry L. Anderson pg 320; DOI: 10.1039/b109915a |
Thionation of bisindole derivatives with P4S10 or elemental sulfur Tomasz Janosik Jan Bergman Birgitta Stensland and Claes Stålhandske pg 330; DOI: 10.1039/b109840c |
N- and O-Alkylation of isoquinolin-1-ones in the Mitsunobu reaction: development of potential drug delivery systems Sandra Ferrer Declan P. Naughton Ifat Parveen and Michael D. Threadgill pg 335; DOI: 10.1039/b109776h |
Reaction of diimines and azines with diphenylcyclopropenone Mohsen Abdel-Motaal Gomaa pg 341; DOI: 10.1039/b109711n |
Photoinduced [2+2] cycloadditions (the Paterno–Bchi reaction) of 1-acetylisatin with enol ethers—regioselectivity, diastereoselectivity and acid catalysed transformations of the spirooxetane products Yan Zhang Jie Xue Yi Gao Hoong-Kun Fun and Jian-Hua Xu pg 345; DOI: 10.1039/b109697d |
Unsymmetrical O-bridged calixarenes derived from tBu-calix[4]arene and p-benzylcalix[4]arene Mohamed Makha Peter J. Nichols Michaele J. Hardie and Colin L. Raston pg 354; DOI: 10.1039/b109625g |
Diastereoselective electrophilic substitution of -amino-substituted benzylic organometallics Ugo Azzena pg 360; DOI: 10.1039/b109633h |
Intramolecular Diels–Alder reaction of cyclopenta-1,3-diene derivatives generated in situ from 4-(pent-4-enyl)cyclopent-2-enone ethylene ketals Masakazu Ohkita Hidetoshi Kawai and Takashi Tsuji pg 366; DOI: 10.1039/b109614a |
Efficient syntheses of 6-prenylcoumarins and linear pyranocoumarins: Total synthesis of suberosin, toddaculin, O-methylapigravin (O-methylbrosiperin), O-methylbalsamiferone, dihydroxanthyletin, xanthyletin and luvangetin Raghao S. Mali Priya P. Joshi Paramjeet Kaur Sandhu and Anita Manekar-Tilve pg 371; DOI: 10.1039/b109597h |
7-Mesityl-2,2-dimethylindan-1-ol: a novel alcohol which serves as both a chiral auxiliary and a protective group for carboxy functions Eiji Koshiishi Tetsutaro Hattori Naoki Ichihara and Sotaro Miyano pg 377; DOI: 10.1039/b109396g |
Regio- and stereoselective synthesis of fluoroalkenes and fluoroalkadienes Masanori Yoshida Daisuke Ota Tsuyoshi Fukuhara Norihiko Yoneda and Shoji Hara pg 384; DOI: 10.1039/b108796g |
Superiority of the carbamoylmethyl ester as an acyl donor for the kinetically controlled amide-bond formation mediated by -chymotrypsin Toshifumi Miyazawa Eiichi Ensatsu Nobuhiro Yabuuchi Ryoji Yanagihara and Takashi Yamada pg 390; DOI: 10.1039/b108735p |
-Chymotrypsin-catalysed segment condensations via the kinetically controlled approach using carbamoylmethyl esters as acyl donors in organic media Toshifumi Miyazawa Eiichi Ensatsu Makoto Hiramatsu Ryoji Yanagihara and Takashi Yamada pg 396; DOI: 10.1039/b108738j |
Flash vacuum pyrolysis over magnesium. Part 1. Pyrolysis of benzylic, other aryl/alkyl and aliphatic halides R. Alan Aitken Philip K. G. Hodgson John J. Morrison and Adebayo O. Oyewale pg 402; DOI: 10.1039/b108663d |
Asymmetric transfer hydrogenation of ketones using amino alcohol and monotosylated diamine derivatives of indane Matthew J. Palmer Jennifer A. Kenny Tim Walsgrove Aparecida M. Kawamoto and Martin Wills pg 416; DOI: 10.1039/b108538g |
Regioselective acylation of 1-hydroxypyrazoles via metalated intermediates Niels Østergaard Niels Skjærbæk Mikael Begtrup and Per Vedsø pg 428; DOI: 10.1039/b107850j |
Reactions of trimethylsilyl-derived iodohydrins with electron-rich -systems Eti Ishai Sarit Shamai and Ben-Ami Feit pg 434; DOI: 10.1039/b105233k |
Phosphabenzenes as electron withdrawing phosphine ligands in catalysis Erin F. DiMauro and Marisa C. Kozlowski pg 439; DOI: 10.1039/b101454o |
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis Gideon Grogan Selena Guilly Ian Jackson Denise McIntyre Reuben Carr Sabine Flitsch and Nicholas Turner pg 4-vii; DOI: 10.1039/b200808b |
Applications of stoichiometric transition metal complexes in organic synthesis Ross Fryatt and Steven D. R. Christie pg 447; DOI: 10.1039/b101946p |
Palladium-catalyzed coupling reaction of acylzirconocene chlorides with hypervalent iodonium salts: synthesis of aryl-substituted ketones Suk-Ku Kang and Seok-Keun Yoon pg 459; DOI: 10.1039/b110983a |
Boronic acid appended azo dyes–colour sensors for saccharides Christopher J. Ward Prakash Patel and Tony D. James pg 462; DOI: 10.1039/b108896c |
Synthesis of 5-arylpyrrolo[1,2-c]pyrimidin-1(2H)-ones Mercedes Álvarez David Fernández and John A. Joule pg 471; DOI: 10.1039/b111142f |
Exploitation of chemical predisposition in synthesis: an approach to the manzamenones Saleh Al-Busafi Jeremy R. Doncaster Michael G. B. Drew Andrew C. Regan and Roger C. Whitehead pg 476; DOI: 10.1039/b110829h |
Synthesis and nucleic-acid-binding properties of sulfamide- and 3-N-sulfamate-modified DNA Kevin J. Fettes Nigel Howard David T. Hickman Steven Adah Mark R. Player Paul F. Torrence and Jason Micklefield pg 485; DOI: 10.1039/b110603c |
A useful enantioselective synthesis of chroman-2-ylmethanol Jean-Yves Goujon Alexis Duval and Bernard Kirschleger pg 496; DOI: 10.1039/b110578g |
Extremely simple and practical synthesis of ()-vertinolide via the Michael addition Kunihiko Takabe Nobuyuki Mase Masaru Nomoto Masanori Daicho Tetsuo Tauchi and Hidemi Yoda pg 500; DOI: 10.1039/b110460h |
Solution-phase combinatorial synthesis using multicomponent Grignard reagents Xifu Liang and Mikael Bols pg 503; DOI: 10.1039/b109952n |
Substitution of -azido ethers with Grignard reagents and its use in combinatorial chemistry Mukulesh Baruah and Mikael Bols pg 509; DOI: 10.1039/b110428b |
Intramolecular addition of acyldiazenecarboxylates onto double bonds in the synthesis of heterocycles José V. Prata Dina-Telma S. Clemente Sundaresan Prabhakar Ana M. Lobo Isabel Mourato (in part) and Paula S. Branco (in part) pg 513; DOI: 10.1039/b110414d |
Synthetic approaches to 1-(2-chlorophenyl)isoquinoline-3-carboxylic acid Yves L. Janin Emmanuel Roulland Arnaud Beurdeley-Thomas Didier Decaudin Claude Monneret and Marie-France Poupon pg 529; DOI: 10.1039/b110301f |
Flash vacuum pyrolysis of stabilised phosphorus ylides. Part 17. Preparation of aliphatic amino acid derived -alkoxycarbonylamino--oxo ylides and pyrolysis to give ,-acetylenic -amino acid and GABA analogues R. Alan Aitken Nazira Karodia Tracy Massil and Robert J. Young pg 533; DOI: 10.1039/b110243e |
Structure of the dimers arising from one-electron electrochemical reduction of pyridinium salts 3,5-disubstituted with electron-withdrawing groups Vincenzo Carelli Felice Liberatore Silvano Tortorella Barbara Di Rienzo and Luigi Scipione pg 542; DOI: 10.1039/b110140b |
3-Hydroxypyrroles and 1H-pyrrol-3(2H)-ones. Part 14. Pyrolysis of oxazolidinylmethylene derivatives of Meldrum's acid – synthesis of N-alkenyl-3-hydroxypyrroles and related reactions Abd El-Aal M. Gaber Gordon A. Hunter and Hamish McNab pg 548; DOI: 10.1039/b109788a |
Control of the reaction between 2-aminobenzothiazoles and Mannich bases. Synthesis of pyrido[2,1-b][1,3]benzothiazoles versus [1,3]benzothiazolo[2,3-b]quinazolines Jairo Quiroga Pedro Hernández Braulio Insuasty Rodrigo Abonía Justo Cobo Adolfo Sánchez Manuel Nogueras and John N. Low pg 555; DOI: 10.1039/b109676a |
Synthesis and chiroptical properties of pseudocolchicine and neocolchicine, novel unnatural regioisomers of colchicine Marino Cavazza Maurizio Zandomeneghi and Francesco Pietra pg 560; DOI: 10.1039/b109075p |
Convergent synthesis of the spiroketal core of the HIV-1 protease inhibitors the didemnaketals Yanxing Jia Xin Li Pingzhen Wang Bin Wu Xuezhi Zhao and Yongqiang Tu pg 565; DOI: 10.1039/b108512n |
Staudinger reactions of unsymmetrical cyclic ketenes: a synthetically useful approach to spiro -lactams and derivatives. Reaction mechanism and theoretical studies Eduardo Alonso Carlos del Pozo and Javier González pg 571; DOI: 10.1039/b103279h |
Professor K. C. Nicolaou* K.C. Nicolaou pg 5-vii; DOI: 10.1039/b200756h |
Perkin 1 Abstracts: Natural Product Synthesis Andrew Gunn Jacqueline E. Milne Marcel de Puit and Duncan McArthur pg 5-xi; DOI: 10.1039/b201458k |
Efficient stereoselective synthesis of peptidomimetics containing hydroxyethylamine dipeptide isosteres utilizing the aza-Payne rearrangement and O, N-acyl transfer reactions Hirokazu Tamamura Tadakazu Hori Akira Otaka and Nobutaka Fujii pg 577; DOI: 10.1039/b200324b |
Arylated pyridines: Suzuki reactions of O-substituted 2,6-dihalogenated-3-hydroxypyridines Glen M. Chapman Stephen P. Stanforth Brian Tarbit and Michael D. Watson pg 581; DOI: 10.1039/b111620g |
The first enantioselective total synthesis of cyclomyltaylane-5-ol and determination of its absolute stereochemistry Hisahiro Hagiwara Hitoshi Sakai Takashi Uchiyama Yoshiaki Ito Noriyuki Morita Takashi Hoshi Toshio Suzuki and Masayoshi Ando pg 583; DOI: 10.1039/b111594b |
Convenient syntheses of 2,3,4,5-tetrahydro-1,4-benzothiazepines, -1,4-benzoxazepines and -1,4-benzodiazepines Alan R. Katritzky Yong-Jiang Xu and Hai-Ying He pg 592; DOI: 10.1039/b111296c |
Synthesis and chemical reactivity of methoxycarbonyl-1,3-dioxinyl(pivaloyl)ketene—a persistent -oxoketene Bianca C. Wallfisch Ferdinand Belaj Curt Wentrup C. Oliver Kappe and Gert Kollenz pg 599; DOI: 10.1039/b111143d |
Studies on tellurium-containing heterocycles. Part 18. Preparation and structure of 2-benzotelluropyrylium salts and 2-benzoselenopyrylium salts Haruki Sashida Kazuo Ohyanagi Mao Minoura and Kin-ya Akiba pg 606; DOI: 10.1039/b111045b |
Synthesis of homochiral amino acid pyrazine and pyrrole analogues of glutamate antagonists Andrew Dinsmore Paul M. Doyle Matthias Steger and Douglas W. Young pg 613; DOI: 10.1039/b110979k |
An approach to 2,3-dihydropyrroles and -iodopyrroles based on 5-endo-dig cyclisations David W. Knight Adele L. Redfern and Jeremy Gilmore pg 622; DOI: 10.1039/b110751h |
A new method for the polymer-supported synthesis of cyclic oligoesters for potential applications in macrocyclic lactone synthesis and combinatorial chemistry Clare L. Ruddick Philip Hodge Anthony Cook and Andrew J. McRiner pg 629; DOI: 10.1039/b110528k |
Arabinose-derived bicyclic amino acids: synthesis, conformational analysis and construction of an v3-selective RGD peptide Francesco Peri Roberta Bassetti Enrico Caneva Luca de Gioia Barbara La Ferla Marco Presta Elena Tanghetti and Francesco Nicotra pg 638; DOI: 10.1039/b110453e |
Novel, cyclic and bicyclic 1,3-diols as catalysts for the diethylzinc addition to aldehydes Ian Sarvary Yiqian Wan and Torbjörn Frejd pg 645; DOI: 10.1039/b110082n |
Facile synthesis of 2-substituted ethyl 2-(2-amino-5-ethoxycarbonylthiazol-4-yl)ethanoates Diana Brikut Frank A. Sløk Christian Rømming and Algirdas akus pg 652; DOI: 10.1039/b110022j |
Synthesis of 2,16- and 4,16-difluoroestradiols and their 11-methoxy derivatives as potential estrogen receptor-binding radiopharmaceuticals Yann Seimbille Hasrat Ali and Johan E. van Lier pg 657; DOI: 10.1039/b110021c |
Ring-opening reactions of cyclopropanes. Part 7. Selenenylation and cyanoselenenylation of ethyl 2,2-dimethoxycyclopropanecarboxylates M. Liliana Graziano M. Rosaria Iesce Flavio Cermola Giovanni Caputo and Fulvio De Lorenzo pg 664; DOI: 10.1039/b109480g |
endo-Selective allylation at the benzylic centre of a Cr(CO)3 complexed aromatic ring Sunil K. Mandal and Amitabha Sarkar pg 669; DOI: 10.1039/b109291j |
,-Didehydroamino acid derivatives with an isoxazolyl or a pyrazolyl moiety: The effect of substituents and reaction conditions on their stereoselective formation from 2H-pyran-2-ones Lidija Vraniar Anton Meden Slovenko Polanc and Marijan Koevar pg 675; DOI: 10.1039/b107624h |
Preparation of novel O-sulfated amino acid building blocks with improved acid stability for Fmoc-based solid-phase peptide synthesis Socorro Vázquez Campos Les P. Miranda and Morten Meldal pg 682; DOI: 10.1039/b107320f |
Stereochemical and electronic features of the [3 + 2] cycloaddition of pentafulvenes with acylnitrones Francis Djapa Kabula Ciamala Jean-Marie Melot Joel Vebrel and Guillaume Herlem pg 687; DOI: 10.1039/b106892j |
A straightforward synthesis of some fused aza-arenes via nucleophilic displacement of a ring hydrogen atom in nitroarenes by aromatic hydrazone anions Koji Uehata Takehiko Kawakami and Hitomi Suzuki pg 696; DOI: 10.1039/b105230f |
Book Reviews pg 703; DOI: 10.1039/b200424k |
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis Gideon Grogan Selena Guilly Ian Jackson Denise McIntyre Reuben Carr Sabine Flitsch and Nicholas Turner pg 6-ix; DOI: 10.1039/b201816k |
New synthesis of ,-diiodoalkynes and capped iodobutadiynes Jaromír Hlavatý Ladislav Kavan and Martin tícha pg 705; DOI: 10.1039/b201360f |
Regioselective reduction of maleimide and citraconimide derivatives: general preparation of 5-hydroxy-1,5-dihydropyrrol-2-one Nobuyuki Mase Toshiki Nishi Masaomi Hiyoshi Kazuhiro Ichihara Junichiro Bessho Hidemi Yoda and Kunihiko Takabe pg 707; DOI: 10.1039/b200729k |
Synthesis of (2E)-4-hydroxy-3-methylbut-2-enyl diphosphate, a key intermediate in the biosynthesis of isoprenoids Jane L. Ward and Michael H. Beale pg 710; DOI: 10.1039/b200712f |
A novel spiroketalization reaction of 1,7-dihydroxyhepta-2,5-diyn-4-ones Koichi Tanaka and Naoyuki Harada pg 713; DOI: 10.1039/b200215a |
Synthesis of the first superstructured chiral corrole Bruno Andrioletti and Eric Rose pg 715; DOI: 10.1039/b200188h |
The preparation of thiophene-based azacryptand Mannich bases Julie D. E. Chaffin John M. Barker and Patrick R. Huddleston pg 717; DOI: 10.1039/b200479h |
Double stereodifferentiation in aldol reactions of pyroglutamic urethane esters Bernard A. Starkmann and Douglas W. Young pg 725; DOI: 10.1039/b200443g |
Synthesis of 2-substituted indolines using sequential Pd-catalyzed processes Hervé J. C. Deboves Christopher Hunter and Richard F. W. Jackson pg 733; DOI: 10.1039/b200163b |
Reactions of acyl chlorides with LiAlHSeH. Preparation of diacyl selenides, diacyl diselenides, selenocarboxylates and cyclic selenoanhydrides Mamoru Koketsu Futoshi Nada Sohma Hiramatsu and Hideharu Ishihara pg 737; DOI: 10.1039/b200147k |
Efficient regioselective synthesis of triheterocyclic compounds: imidazo[2,1-b]benzothiazoles, pyrimido[2,1-b]benzothiazolones and pyrimido[2,1-b]benzothiazoles Cyrille Landreau David Deniaud Michel Evain Alain Reliquet and Jean-Claude Meslin pg 741; DOI: 10.1039/b111639h |
Dendritic encapsulation of amino acid–metal complexes. Synthesis and studies of dendron-functionalized L-tyrosine–metal (ZnII, CoII) complexes Thatavarathy Rama Krishna and Narayanaswamy Jayaraman pg 746; DOI: 10.1039/b110188a |
Application of [5+2] cycloaddition toward the functionalized bicyclo[4.3.1]decane ring system: synthetic study of phomoidride B (CP-263,114) Naoki Ohmori pg 755; DOI: 10.1039/b110607b |
Synthetic and mechanistic study of the acid-promoted aromatisation of the Diels–Alder adduct: 6,7-dimethoxy-1-(4-pyridyl)-1,4-epoxytetrahydronaphthalene-2,3-dicarboxylate Masakatsu Sugahara Yasunori Moritani Tooru Kuroda Kazuhiko Kondo and Tatsuzo Ukita pg 768; DOI: 10.1039/b110265f |
Tandem sigmatropic shifts in [4 + 2] cycloaddition reactions of 1,3-diazabuta-1,3-dienes with butadienylketene: synthesis of pyrimidinone derivatives Arun K. Sharma S. Jayakumar Maninder S. Hundal and Mohinder P. Mahajan pg 774; DOI: 10.1039/b109922c |
A facile and simple entry into isodideoxynucleosides Angshuman Chattopadhyay and Avinash Salaskar pg 785; DOI: 10.1039/b109785g |
Synthesis of quinoxaline derivatives from substituted acetanilides through intramolecular quaternization reactions Sonia de Castro Roberto Chicharro and Vicente J. Arán pg 790; DOI: 10.1039/b109725c |
Modular fluorescence sensors for saccharides Susumu Arimori Michael L. Bell Chan S. Oh Karine A. Frimat and Tony D. James pg 803; DOI: 10.1039/b108998f |
Insights on the synthesis and organisational phenomena of twisted pyrazine–pyridine hybrids Fenton Heirtzler Markus Neuburger and Klaus Kulike pg 809; DOI: 10.1039/b107751a |
An efficient synthesis of the four mono methylated isomers of (+)-catechin including the major metabolites and of some dimethylated and trimethylated analogues through selective protection of the catechol ring Cécile Cren-Olivé Stéphane Lebrun and Christian Rolando pg 821; DOI: 10.1039/b107340k |
Novel glucocorticoid antedrugs possessing a 21-(-lactone) ring Richard M. Angell Keith Biggadike Rosanne M. Farrell Stephen S. Flack Ashley P. Hancock Wendy R. Irving Sean M. Lynn and Panayiotis A. Procopiou pg 831; DOI: 10.1039/b200190j |
Perkin 1 Abstracts: Solid Phase Organic Synthesis Andrew Gunn Stephen McAteer and Marcel de Puit pg 7-vii; DOI: 10.1039/b202398a |
Synthetic receptors for carboxylic acids and carboxylates Richard J. Fitzmaurice Graham M. Kyne David Douheret and Jeremy D. Kilburn pg 841; DOI: 10.1039/b009041g |
Alkali metal ion selectivities of podands that form pseudo-cyclic structures by intramolecular hydrogen bonding Yoichi Habata Yoji Fukuda Sadatoshi Akabori and Jerald S. Bradshaw pg 865; DOI: 10.1039/b201525k |
Highly enantioselective epoxidation of unfunctionalized olefins catalyzed by a novel recyclable chiral poly-salen–Mn(III) complex Yuming Song Xiaoquan Yao Huilin Chen Guizhi Pan Xinquan Hu and Zhuo Zheng pg 870; DOI: 10.1039/b201294b |
The use of -allyltricarbonyliron lactone complexes in the synthesis of the resorcylic macrolides - and -zearalenol Svenja Burckhardt and Steven V. Ley pg 874; DOI: 10.1039/b201164f |
Olefination of aromatic ketones: synthesis of mono- and dihaloalkenes Vasily N. Korotchenko Alexey V. Shastin Valentine G. Nenajdenko and Elisabeth S. Balenkova pg 883; DOI: 10.1039/b201131j |
Resolution and configurational assignment of 3,4,5,6-tetrahydro-2-methyl-2,6-methano-2H-1-benzoxocine derivatives Tibor Kurtán Eszter Baitz-Gács Zsuzsa Májer Attila Bényei and Sándor Antus pg 888; DOI: 10.1039/b200751g |
Total synthesis of bisabolane sesquiterpenoids, -bisabol-1-one, curcumene, curcuphenol and elvirol: utility of catalytic enamine reaction in cyclohexenone synthesis Hisahiro Hagiwara Tomoyuki Okabe Hiroki Ono Vijayendra P. Kamat Takashi Hoshi Toshio Suzuki and Masayoshi Ando pg 895; DOI: 10.1039/b200629b |
Atroposelectivity in the electrophilic substitution reactions of laterally lithiated and silylated tertiary amides Jonathan Clayden Jennifer H. Pink Neil Westlund and Christopher S. Frampton pg 901; DOI: 10.1039/b200358a |
Synthesis of cholic acid-based molecular receptors: head-to-head cholaphanes Pramod S. Pandey Roopali Rai and Rhiddi B. Singh pg 918; DOI: 10.1039/b200320c |
Synthesis of ABE tricyclic analogues of methyllycaconitine using a Wacker oxidation–aldol strategy to append the B ring to the AE fragment David Barker Margaret A. Brimble Malcolm McLeod G. Paul Savage and David J. Wong pg 924; DOI: 10.1039/b200073n |
Synthesis, characterisation and application of lanthanide cyclen complexes in organic synthesis Andrei S. Batsanov James I. Bruce Thota Ganesh Paul J. Low Ritu Kataky Horst Puschmann and Patrick G. Steel pg 932; DOI: 10.1039/b111628b |
Pigments of fungi. Part 68. Synthesis and absolute configuration of thysanone Christopher D. Donner and Melvyn Gill pg 938; DOI: 10.1039/b111446h |
Enantioselective total synthesis of vicenistatin, a novel 20-membered macrocyclic lactam antitumor antibiotic Yoshitaka Matsushima Hiroaki Itoh Takuya Nakayama Sayo Horiuchi Tadashi Eguchi and Katsumi Kakinuma pg 949; DOI: 10.1039/b111146a |
Stereoselectivity in ring-closing olefin metathesis (RCM) of tethered dihexenoyl derivatives Mitsuhiro Arisawa Hiroaki Kaneko Atsushi Nishida and Masako Nakagawa pg 959; DOI: 10.1039/b111122c |
Synthesis of 2,5-dihydrofurans via alkylidene carbene insertion reactions Louise F. Walker Ahmed Bourghida Stephen Connolly and Martin Wills pg 965; DOI: 10.1039/b111097g |
Molecular recognition of modified nucleobases. Self-complementarity and base-pairing of betainic guanine model compounds Andreas Schmidt Nikoloz Kobakhidze and Markus Karl Kindermann pg 982; DOI: 10.1039/b110318k |
A facile route to poly[1-(2,4,6-trichlorophenyl)-1H-1,2,4-triazol-5-yl]alkane derivatives Quanrui Wang Haiyan Yang Yi Liu Zongbiao Ding and Fenggang Tao pg 991; DOI: 10.1039/b110059a |
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis Gideon Grogan Selena Guilly Ian Jackson Denise McIntyre Reuben Carr Sabine Flitsch and Nicholas Turner pg 8-vii; DOI: 10.1039/b202864f |
Polyene natural products Carl Thirsk and Andrew Whiting pg 999; DOI: 10.1039/b109741p |
The simultaneous use of immobilised reagents for the one-pot conversion of alcohols to carboxylic acids Kosuke Yasuda and Steven V. Ley pg 1024; DOI: 10.1039/b201776h |
An exceptionally simple and catalytic method for regeneration of carbonyl functionality from the corresponding 1,3-oxathiolanes Ejabul Mondal Priti Rani Sahu Gopal Bose and Abu T. Khan pg 1026; DOI: 10.1039/b110305a |
Synthesis and in vitro enzyme activity of an oxa analogue of azi-DAP Russell J. Cox Jeremy Durston and David I. Roper pg 1029; DOI: 10.1039/b201727j |
Self-terminating, oxidative radical cyclizations of medium-sized cycloalkynones with inorganic and organic oxygen-centered radicals of type XO: the reaction pathway depends on the nature of X Uta Wille and Christian Jargstorff pg 1036; DOI: 10.1039/b201672a |
A convenient preparation of several N-linked glycoamino acid building blocks for efficient solid-phase synthesis of glycopeptides Jeroen van Ameijde H. Bauke Albada and Rob M. J. Liskamp pg 1042; DOI: 10.1039/b201296k |
Synthesis of enantiomerically pure divinyl- and diallylcarbinols Bernd Schmidt and Holger Wildemann pg 1050; DOI: 10.1039/b200976e |
Total synthesis of naamine C and pyronaamidine, antitumor marine imidazole alkaloids Seikou Nakamura Ikuo Kawasaki Miki Kunimura Miyuki Matsui Yoko Noma Masayuki Yamashita and Shunsaku Ohta pg 1061; DOI: 10.1039/b200845a |
Synthesis and biological evaluation of a PtdIns(4,5)P2 and a phosphatidic acid affinity matrix Ze-Yi Lim Jan W. Thuring Andrew B. Holmes Maria Manifava and Nicholas T. Ktistakis pg 1067; DOI: 10.1039/b200585a |
Diastereoselective addition of chiral azomethine ylides to cyclic ,-unsaturated N-enoylbornanesultams Staffan Karlsson and Hans-Erik Högberg pg 1076; DOI: 10.1039/b200579d |
Approaches to the synthesis of (2R,3S)-2-hydroxymethylpyrrolidin-3-ol (CYB-3) and its C(3) epimer: a cautionary tale Alison N. Hulme and Karen S. Curley pg 1083; DOI: 10.1039/b200415a |
Novel uridin-2-yl carbamates: synthesis, incorporation into oligodeoxyribonucleotides, and remarkable fluorescence properties of 2-pyren-1-ylmethylcarbamate Vladimir A. Korshun Dmitry A. Stetsenko and Michael J. Gait pg 1092; DOI: 10.1039/b111434b |
Intramolecular acceleration effect of a tosylamide group on the electrochemical oxidation of N--silylalkyl amides Tohru Kamada and Akira Oku pg 1105; DOI: 10.1039/b111106j |
Screening of yeast species for the stereo-selective reduction of bicyclo[2.2.2]octane-2,6-dione Adriana L. Botes Daniel Harvig Martha S. van Dyk Ian Sarvary Torbjörn Frejd Mikael Katz Bärbel Hahn-Hägerdal and Marie F. Gorwa-Grauslund pg 1111; DOI: 10.1039/b111064k |
Regiocontrolled synthesis of the macrocyclic polyamine alkaloid ()-lunarine, a time-dependent inhibitor of trypanothione reductase Chris J. Hamilton Alan H. Fairlamb and Ian M. Eggleston pg 1115; DOI: 10.1039/b110149h |
Synthesis of glycero amino acid-based surfactants. Part 2. Lipase-catalysed synthesis of 1-O-lauroyl-rac-glycero-3-O-(N-acetyl-L-amino acid) and 1,2-di-O-lauroyl-rac-glycero-3-O-(N-acetyl-L-amino acid) derivatives Carmen Morán María Rosa Infante and Pere Clapés pg 1124; DOI: 10.1039/b200577h |
Electrochemical synthesis of a pyridinium-conjugated assembly based on nucleophilic substitution of oligothiophene -radical cation Yi Li Kaori Kamata Tadashi Kawai Jiro Abe and Tomokazu Iyoda pg 1135; DOI: 10.1039/b200738j |
Perkin 1 Abstracts: Solid Phase Organic Synthesis Fabrice Anizon Jennifer Delaney Andrew Gunn Hassan Mamdani Catherine McCusker Fiona McKerlie and Tanya Wildman pg 9-v; DOI: 10.1039/b203347j |
Recent developments in the chemistry of dihydropyridines Rodolfo Lavilla pg 1141; DOI: 10.1039/b101371h |
Tin(II) chloride mediated allylation of aldimines generated in situ with allylstannane in water Takahiko Akiyama and Yuji Onuma pg 1157; DOI: 10.1039/b202486a |
The reaction of dialkoxytitanacyclopropanes and dialkoxytitanacyclopropenes with carbon dioxide Yvan Six pg 1159; DOI: 10.1039/b201527g |
Deoxygenation of tertiary and secondary alcohols ROH by thiol-catalysed radical-chain redox decomposition of derivatives ROCH2X to give RH and XCHO Hai-Shan Dang and Brian P. Roberts pg 1161; DOI: 10.1039/b202411j |
Distorted electron acceptors: an unexpected reaction involving tetramethyl-TCNQ Norman A. Bell David J. Crouch Lawrence R. H. High Derek J. Simmonds Simon J. Coles and Michael B. Hursthouse pg 1171; DOI: 10.1039/b201862b |
Synthesis, X-ray crystal structures and Horner–Wittig addition reactions of some protected -aminophosphine oxides Neil Feeder David J. Fox Jonathan A. Medlock and Stuart Warren pg 1175; DOI: 10.1039/b201680j |
Parallel synthesis of new phenylalanino-2-(phenylthio)pyrrolidin-3-one scaffold-based analogues Gilles Quéléver Martin Bouygues and Jean-Louis Kraus pg 1181; DOI: 10.1039/b201147f |
Synthesis and investigation of L-fuco- and D-glucurono-azafagomine Henrik H. Jensen Astrid Jensen Rita G. Hazell and Mikael Bols pg 1190; DOI: 10.1039/b200884j |
Synthesis of (1S,2R)-1-phenyl-2-[(S)-1-aminoalkyl]-N,N-diethylcyclopropanecarboxamides as novel NMDA receptor antagonists having a unique NMDA receptor subtype selectivity Yuji Kazuta Ryuichi Tsujita Shigeo Uchino Noriko Kamiyama Daisuke Mochizuki Kanako Yamashita Yutaka Ohmori Akitake Yamashita Tamotsu Yamamoto Shinich Kohsaka Akira Matsuda and Satoshi Shuto pg 1199; DOI: 10.1039/b111540p |
Structural effects on sigmatropic shifts in heteroaromatic allyl ethers Nuna C. P. Araújo Pedro M. M. Barroca Jamie F. Bickley Amadeu F. Brigas M. Lurdes S. Cristiano Robert A. W. Johnstone Rui M. S. Loureiro and Paula C. A. Pena pg 1213; DOI: 10.1039/b102674g |
Book Reviews pg 1220; DOI: 10.1039/b202565p |
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis Gideon Grogan Selena Guilly Ian Jackson Denise McIntyre Reuben Carr Sabine Flitsch and Nicholas Turner pg 10-vii; DOI: 10.1039/b203807m |
Efficient and chemoselective cleavage of TBS ethers by a sub-stoichiometric amount of decaborane Yeon Joo Jeong Ji Hee Lee Eun Soo Park and Cheol Min Yoon pg 1223; DOI: 10.1039/b201794f |
Synthesis of a linear bis-porphyrin with a Ru(phen)22+-complexed 2,2-bipyridine spacer James I. Bruce Jean-Claude Chambron Philipp Kölle and Jean-Pierre Sauvage pg 1226; DOI: 10.1039/b202407c |
Synthesis of fluorinated 2-phenyl-4-quinolones from pyrrole-2,3-diones V. V. Ramana Rao and Curt Wentrup pg 1232; DOI: 10.1039/b202128e |
Reactions of 1,2,3-dithiazoles with halogenated malononitriles Irene C. Christoforou Panayiotis A. Koutentis and Charles W. Rees pg 1236; DOI: 10.1039/b202038f |
Synthesis and evaluation of sulfonium analogues of isofucofagomine as glycosidase inhibitors Víctor Ulgar José G. Fernández-Bolaños and Mikael Bols pg 1242; DOI: 10.1039/b202021c |
Solid phase synthesis of C2,N6-disubstituted adenosine analogues Boris Rodenko Martin J. Wanner and Gerrit-Jan Koomen pg 1247; DOI: 10.1039/b201943d |
Aminolysis of cyclic thioxocarbonate of (R,R)-di-tert-butyl tartrate: efficient access to thio- and thiolcarbamates Ludovic Faissat Claude Chavis Jean-Louis Montéro and Marc Lucas pg 1253; DOI: 10.1039/b201691e |
Novel heterocycles containing the pyrazole unit Jan Svtlík and Tibor Liptaj pg 1260; DOI: 10.1039/b201529n |
Synthesis and analysis of peptide nucleic acid oligomers using Fmoc/acyl-protected monomers Györgyi Kovács Zoltán Timár Zoltán Kupihár Zoltán Kele and Lajos Kovács pg 1266; DOI: 10.1039/b201297a |
Synthesis of S-thioacyl dithiophosphates, efficient and chemoselective thioacylating agents Leszek Doszczak and Janusz Rachon pg 1271; DOI: 10.1039/b201233b |
Solvent-free chelation-assisted hydroacylation of olefin by rhodium(I) catalyst under microwave irradiation André Loupy Saber Chatti Sarah Delamare Dae-Yon Lee Jong-Hwa Chung and Chul-Ho Jun pg 1280; DOI: 10.1039/b200442a |
Synthesis of chiral organotin reagents: synthesis of enantiomerically enriched bicyclo[2.2.1]hept-2-yl tin hydrides from camphor. X-Ray crystal structures of (dimethyl)[(1R,2S,4R)-1,7,7-trimethylbicyclo[2.2.1]hept-2-yl]tin chloride and methyl(phenyl)bis[(1R,2S,4R)-1,7,7-trimethylbicyclo[2.2.1]hept-2-yl]stannane Madeleine Helliwell Eric J. Thomas and Linda A. Townsend pg 1286; DOI: 10.1039/b200317c |
Investigation of the base promoted tandem syn-elimination–Favorskii rearrangement of levoglucosan sulfonates Lene Muldgaard Ib B. Thomsen Rita G. Hazell and Mikael Bols pg 1297; DOI: 10.1039/b200064b |
In vitro fluorine-19 nuclear magnetic resonance study of the liberation of antitumor nitrogen mustard from prodrugs Frédéric Schmidt and Claude Monneret pg 1302; DOI: 10.1039/b111549a |
Efficient synthesis of -substituted -haloenones by rhodium(II)-catalyzed and thermal reactions of iodonium ylides Yong Rok Lee and Yong Ug Jung pg 1309; DOI: 10.1039/b111206f |
Indium-mediated diastereoselective allylation reactions: preparation of -hydroxy and -amino acids Jung Gyu Lee Kyung Il Choi Ae Nim Pae Hun Yeong Koh Yonghan Kang and Yong Seo Cho pg 1314; DOI: 10.1039/b110505c |
A convenient general synthesis of 3-substituted 2H-chromene derivatives Perry T Kaye and Xolani W. Nocanda pg 1318; DOI: 10.1039/b201827f |
Perkin 1 Abstracts: Natural Product Synthesis Andrew Gunn Stephen McAteer Jacqueline E. Milne and Marcel de Puit pg 11-ix; DOI: 10.1039/b204498f |
Boron acids as protective agents and catalysts in synthesis Peter J. Duggan and Edward M. Tyndall pg 1325; DOI: 10.1039/b006767i |
Rapid and convergent assembly of the polycyclic framework assigned to the cytotoxic marine alkaloid halitulin Martin G. Banwell Andrew M. Bray Alison J. Edwards and David J. Wong pg 1340; DOI: 10.1039/b111401h |
Synthetic studies on CP-225,917 and CP-263,114: concise synthesis of the bicyclic core using an intramolecular Mukaiyama aldol reaction Alan Armstrong Trevor J. Critchley Marie-Edith Gourdel-Martin Richard D. Kelsey and Andrew A. Mortlock pg 1344; DOI: 10.1039/b202752f |
Synthesis of pseudoxazolones and their inhibition of the 3C cysteine proteinases from hepatitis A virus and human rhinovirus-14 Yeeman K. Ramtohul Nathaniel I. Martin Lara Silkin Michael N. G. James and John C. Vederas pg 1351; DOI: 10.1039/b202643k |
Intramolecular Michael-type addition of azadienes to 1,4-naphthoquinones instead of Aza-Diels–Alder cycloaddition: a synthesis of ascididemin Juan M. Cuerva Diego J. Cárdenas and Antonio M. Echavarren pg 1360; DOI: 10.1039/b202555h |
Quinolizine-2,4-diones by reversible dimerisation 2-pyridylketenes Carsten Plüg Arvid Kuhn and Curt Wentrup pg 1366; DOI: 10.1039/b202523j |
Preparation of (+)-nemorensic acid and approaches to nemorensine using the partial reduction of electron deficient furans Timothy J. Donohoe Jean-Baptiste Guillermin and Daryl S. Walter pg 1369; DOI: 10.1039/b202514k |
Carbohydrate-derived thiols as protic polarity-reversal catalysts for enantioselective radical-chain reactions Yudong Cai Brian P. Roberts and Derek A. Tocher pg 1376; DOI: 10.1039/b202022j |
Stereocontrolled synthesis of acyclic terpenoids viaN-ylide [2,3]rearrangement of ammonium salts with the stereodefined isoprene unit Kiyoshi Honda Masayuki Tabuchi Hiroki Kurokawa Masatoshi Asami and Seiichi Inoue pg 1387; DOI: 10.1039/b201304e |
Synthesis of unsymmetrically substituted meso-phenylporphyrins by Suzuki cross coupling reactions Baolu Shi and Ross W. Boyle pg 1397; DOI: 10.1039/b201622b |
Elemental iodine catalyzed [4 + 2] cycloaddition reactions of o-quinomethanes: an efficient synthesis of trans-fused pyrano[3,2-c]benzopyrans Jhillu Singh Yadav Basi V. Subba Reddy C. Venkateswara Rao and K. Vishweshwar Rao pg 1401; DOI: 10.1039/b200193b |
Symmetrical and inherently chiral water-soluble calix[4]arenes bearing dihydroxyphosphoryl groups Maxim A. Tairov Myroslav O. Vysotsky Olga I. Kalchenko Vladimir V. Pirozhenko and Vitaly I. Kalchenko pg 1405; DOI: 10.1039/b110691k |
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis Gideon Grogan Selena Guilly Ian Jackson Denise McIntyre Reuben Carr Sabine Flitsch and Nicholas Turner pg 12-vii; DOI: 10.1039/b204941b |
The first isolation and characterization of sulfonylbuta-1,3-diynes Mitsuhiro Yoshimatsu Kasumi Oh-Ishi Genzoh Tanabe and Osamu Muraoka pg 1413; DOI: 10.1039/b203913n |
Synthesis and light absorption/emission properties of novel bis-squaraine dyes with extensively conjugated -electron systems Shigeyuki Yagi Shin Murayama Yutaka Hyodo Yoshihiko Fujie Msahiko Hirose and Hiroyuki Nakazumi pg 1417; DOI: 10.1039/b203793a |
The role of the carbonyl group in the intermolecular 1,3-cycloaddition of azido(2-heteroaryl)methanones with activated olefins Paolo Zanirato pg 1420; DOI: 10.1039/b203577d |
Carbanion induced synthesis of annulated unsymmetrical biaryls through ring transformation of 2H-pyran-2-one Vishnu Ji Ram Nidhi Agarwal Abhishek S. Saxena Farhanullah Ashoke Sharon and Prakas R. Maulik pg 1426; DOI: 10.1039/b203544h |
A new entry to 9-azabicyclo[3.3.1]nonanes using radical translocation/cyclisation reactions of 2-(but-3-ynyl)-1-(o-iodobenzoyl)piperidines Tatsunori Sato Taro Yamazaki Yumi Nakanishi Jun-ichi Uenishi and Masazumi Ikeda pg 1438; DOI: 10.1039/b203243k |
Towards complete stereochemical control: complementary methods for the synthesis of six diastereoisomeric monosaccharide mimetics Robert Hodgson Tahir Majid and Adam Nelson pg 1444; DOI: 10.1039/b202890e |
Synthesis of some 3,4-dihydro-2H-benzo[f]pyrano[2,3-h]chromen-6-one derivatives Demetrios N. Nicolaides Daman R. Gautam Konstantinos E. Litinas and Theodora Papamehael pg 1455; DOI: 10.1039/b202640f |
Tributyltin hydride-mediated radical cyclisation of carbonyls to form functionalised oxygen and nitrogen heterocycles Jon Bentley Paul A. Nilsson and Andrew F. Parsons pg 1461; DOI: 10.1039/b202077g |
Chemical reactivity of hydroxymethylnaphthols: hetero-Diels–Alder products of o-naphthoquinomethides derived from 2- and 3-hydroxymethylnaphthols Muhammad Ashram David O. Miller and Paris E. Georghiou pg 1470; DOI: 10.1039/b200893a |
Synthesis of (E)- and (Z)-29-methylidyne-2,3-oxidosqualene derivatives as inhibitors of liver and yeast oxidosqualene cyclase Maurizio Ceruti Franca Viola Gianni Balliano Paola Milla Giorgio Roma Giancarlo Grossi and Flavio Rocco pg 1477; DOI: 10.1039/b200888m |
Reaction of -carbanion of imines with N-tosylimines: a facile route to -aminoaldehydes and 1,3-diamines Xue-Long Hou Yu-Mei Luo Ke Yuan and Li-Xin Dai pg 1487; DOI: 10.1039/b200198e |
Direct NH-aziridination of ,-unsaturated ketones Jiaxi Xu and Peng Jiao pg 1491; DOI: 10.1039/b200046f |
Nitrone dipolar cycloaddition routes to piperidines and indolizidines. Part 9. Formal synthesis of (–)-pinidine and total synthesis of (–)-histrionicotoxin, (+)-histrionicotoxin and (–)-histrionicotoxin 235A Edwin C. Davison Martin E. Fox Andrew B. Holmes Stephen D. Roughley Catherine J. Smith Geoffrey M. Williams John E. Davies Paul R. Raithby Joseph P. Adams Ian T. Forbes Neil J. Press and Mervyn J. Thompson pg 1494; DOI: 10.1039/b200328g |
Efficient synthesis of functionalized 3H-pyrrolo[1,2-a]indoles Issa Yavari Mehdi Adib and Mohammad H. Sayahi pg 1517; DOI: 10.1039/b204433c |
Catalysis by ionic liquids: solvent-free efficient transthioacetalisation of acetals by molten tetrabutylammonium bromide Brindaban C. Ranu Arijit Das and Sampak Samanta pg 1520; DOI: 10.1039/b204363g |
High surface area polystyrene resin-supported Pt catalysts in room temperature solventless octene hydrosilylation using methyldichlorosilane Robert Drake David C. Sherrington and Steven J. Thomson pg 1523; DOI: 10.1039/b203899d |
Conversion of tetrazoles into hydrazonoyl chlorides. Novel donor–dithiazolium interactions Charles W. Rees Sivaprasad Sivadasan Andrew J. P. White and David J. Williams pg 1535; DOI: 10.1039/b202211g |
Synthesis of 1,3,4-thiadiazole oligomers Van-Duc Le Charles W. Rees and Sivaprasad Sivadasan pg 1543; DOI: 10.1039/b203705j |
Palladium(II) complex-catalysed enantioselective benzoylation of alcohols using carbon monoxide and an organobismuth(V) compound Tomochika Iwata Yoshihiro Miyake Yoshiaki Nishibayashi and Sakae Uemura pg 1548; DOI: 10.1039/b203465d |
Conversion of (Z)-1,4-dihydroxyalk-2-enes into 2,5-dihydrofurans and of alkane-1,4-diols into tetrahydrofurans via acid-catalysed cyclisation of the monoisoureas formed by their copper(I)-mediated reactions with dicyclohexylcarbodiimide Michael G. Duffy and David H. Grayson pg 1555; DOI: 10.1039/b203389p |
Expeditious preparation of various 9-6a,10a cis and trans 2-substituted tetrahydrocannabinoids Jean-Yves Goujon Françoise Zammattio and Bernard Kirschleger pg 1564; DOI: 10.1039/b203366f |
Synthesis of diselenadiazafulvalenes and influence of steric strain on their anodic behavior Zdenko asar Ivan Leban Alenka Majcen-Le Maréchal and Dominique Lorcy pg 1568; DOI: 10.1039/b203317h |
Reaction of 5-halo-1,2,3-thiadiazoles with arylenediamines as a new approach to tricyclic 1,3,6-thiadiazepines Natalya N. Volkova Evgeniy V. Tarasov Luc Van Meervelt Suzanne Toppet Wim Dehaen and Vasiliy A. Bakulev pg 1574; DOI: 10.1039/b203072a |
Carotenoids and related polyenes. Part 8. Total synthesis of optically active mytiloxanthin applying the stereoselective rearrangement of tetrasubstituted epoxide Chisato Tode Yumiko Yamano and Masayoshi Ito pg 1581; DOI: 10.1039/b201228f |
Synthesis of pyrazole and pyrimidine Trger's-base analogues Rodrigo Abonia Andrea Albornoz Hector Larrahondo Jairo Quiroga Braulio Insuasty Henry Insuasty Angelina Hormaza Adolfo Sánchez and Manuel Nogueras pg 1588; DOI: 10.1039/b200862a |
Novel photoadditions of tertiary amines to the -position of ,-unsaturated ,-epoxy nitriles Keitaro Ishii Satoshi Hakamada Mayumi Nagano Masahiro Noji Shigeo Sugiyama Masashi Kotera and Masanori Sakamoto pg 1592; DOI: 10.1039/b110372e |
Book Reviews pg 1599; DOI: 10.1039/b205252k |
Perkin 1 Abstracts: Natural Product Synthesis Andrew Gunn Stephen McAteer Jacqueline E. Milne and Marcel de Puit pg 14-x; DOI: 10.1039/b205788n |
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis Gideon Grogan Selena Guilly Ian Jackson Denise McIntyre Reuben Carr Sabine Flitsch and Nicholas Turner pg 14-vii; DOI: 10.1039/b206029a |
Annulenes, 1980–2000 Robert D. Kennedy Douglas Lloyd and Hamish McNab pg 1601; DOI: 10.1039/b109576p |
A chemoenzymatic synthesis of the styryllactone (+)-goniodiol from naphthalene Martin G. Banwell Mark J. Coster Ochitha P. Karunaratne and Jason A. Smith pg 1622; DOI: 10.1039/b205230j |
Synthesis and biological evaluation of phospholane and dihydrophosphole analogues of the glutamate receptor agonist AP4 Stuart J. Conway Jacqueline C. Miller Andrew D. Bond Barry P. Clark and David E. Jane pg 1625; DOI: 10.1039/b204891d |
Unprecedented 1,3-dipolar cycloaddition of azomethine ylides to ester carbonyl Mikhail S. Novikov Igor V. Voznyi Alexander F. Khlebnikov Jürgen Kopf and Rafael R. Kostikov pg 1628; DOI: 10.1039/b204464a |
Desymmetrisation of meso difuryl alcohols, diols and their derivatives: complementary directed and undirected asymmetric dihydroxylation reactions Robert Hodgson Tahir Majid and Adam Nelson pg 1631; DOI: 10.1039/b204904j |
Streptomyces coelicolor phosphopantetheinyl transferase: a promiscuous activator of polyketide and fatty acid synthase acyl carrier proteins Russell J. Cox John Crosby Oliver Daltrop Frank Glod Malgorzata E. Jarzabek Thomas P. Nicholson Michelle Reed Thomas J. Simpson Leah H. Smith Florilène Soulas Anna E. Szafranska and James Westcott pg 1644; DOI: 10.1039/b204633b |
Synthesis of chiral oxazolidin-2-ones from N-alkoxycarbonyl amino epoxides: a computational study F. Javier Casado-Bellver M. Eugenia González-Rosende Amparo Asensio J. Miquel Jordá-Gregori Angeles Alvarez-Sorolla José Sepúlveda-Arques Mario Orena and Roberta Galeazzi pg 1650; DOI: 10.1039/b203702e |
Synthesis and antiviral evaluation of novel conformationally locked nucleosides and masked 5-phosphate derivatives thereof Torsten Bryld Marianne H. Sørensen Poul Nielsen Troels Koch Claus Nielsen and Jesper Wengel pg 1655; DOI: 10.1039/b203484k |
Synthesis of tetrasubstituted pyridines by the acid-catalysed Bohlmann–Rahtz reaction Mark C. Bagley Christian Brace James W. Dale Maren Ohnesorge Nathan G. Phillips Xin Xiong and Justin Bower pg 1663; DOI: 10.1039/b203397f |
N–H Insertion reactions of rhodium carbenoids. Part 3. The development of a modified Bischler indole synthesis and a new protecting-group strategy for indoles Katherine E. Bashford Anthony L. Cooper Peter D. Kane Christopher J. Moody Sendogagounder Muthusamy and Elizabeth Swann pg 1672; DOI: 10.1039/b202666j |
Novel trichloroindolizine derivatives via intramolecular acylation of a bis(chloroacyl)bipyridine Najat Sam Sghir Elkadiri Hubert Le Bozec Loic Toupet Maria Daoudi Najib Bitit Taibi Ben Hadda and Pierre H. Dixneuf pg 1688; DOI: 10.1039/b202616n |
Studies towards the total synthesis of solanoeclepin A: synthesis of the 7-oxabicyclo[2.2.1]heptane moiety and attempted seven-membered ring formation Jorg C. J. Benningshof Richard H. Blaauw Angeline E. van Ginkel Jan H. van Maarseveen Floris P. J. T. Rutjes and Henk Hiemstra pg 1693; DOI: 10.1039/b201987f |
Studies towards the total synthesis of solanoeclepin A: synthesis and potato cyst nematode hatching activity of analogues containing the tetracyclic left-hand substructure Jorg C. J. Benningshof Maarten IJsselstijn Sabine R. Wallner Anne L. Koster Richard H. Blaauw Angeline E. van Ginkel Jean-François Brière Jan H. van Maarseveen Floris P. J. T. Rutjes and Henk Hiemstra pg 1701; DOI: 10.1039/b202020n |
Thioester analogues of peptidoglycan fragment MurNAc-L-Ala--D-Glu as substrates for peptidoglycan hydrolase MurNAc-L-Ala amidase Ross L. Harding Joanne Henshaw Joannah Tilling and Timothy D. H. Bugg pg 1714; DOI: 10.1039/b200921h |
Synthesis and binding properties of chiral macrocyclic barbiturate receptors: application to nitrile oxide cyclizations Brian S. Rasmussen Unai Elezcano and Troels Skrydstrup pg 1723; DOI: 10.1039/b110865b |
Perkin 1 Abstracts: Natural Product Synthesis Andrew Gunn Stephen McAteer Jacqueline E. Milne and Marcel de Puit pg 15-vii; DOI: 10.1039/b206710m |
The emergence of the cyclopentenone prostaglandins as important, biologically active compounds Stanley M. Roberts M. Gabriella Santoro and Eugene S. Sickle pg 1735; DOI: 10.1039/b110043m |
C-Glycoside formation via Lewis acid promoted reaction of O-glycosylimidates with pyrroles David J. Armitt Martin G. Banwell Craig Freeman and Christopher R. Parish pg 1743; DOI: 10.1039/b205690a |
Acid catalysed rearrangement of a spiroketal enol ether. An easy synthesis of chrycorin Biao-Lin Yin Yikang Wu and Yu-Lin Wu pg 1746; DOI: 10.1039/b205229f |
Partial reduction of 3-heteroatom substituted 2-furoic acids: the role of an ortho group in viability and stereoselectivity Timothy J. Donohoe Andrew A. Calabrese Jean-Baptiste Guillermin Christopher. S. Frampton and Daryl Walter pg 1748; DOI: 10.1039/b203437a |
The [2,3] sigmatropic rearrangement of N-benzyl-O-allylhydroxylamines Stephen G. Davies John F. Fox Simon Jones Anne J. Price Miguel A. Sanz Thomas G. R. Sellers Andrew D. Smith and Fátima C. Teixeira pg 1757; DOI: 10.1039/b205323n |
Microwave assisted facile synthesis of Elvirol, Curcuphenol and Sesquichamaenol using Montmorillonite K-10 clay in dry media Vasundhara Singh Anupam Khurana Irvinder Kaur Varinder Sapehiyia Goverdhan L. Kad and Jasvinder Singh pg 1766; DOI: 10.1039/b204509p |
Heteroaryl radicals. Part 1. Synthesis of linear pyridine-fused ring systems by endo-selective 2-pyridyl radical cyclizations Sarbendu Maiti Basudeb Achari Ranjan Mukhopadhyay and Asish Kr. Banerjee pg 1769; DOI: 10.1039/b204436f |
NMR characterisation of five isomeric ,-diformyl-meso-tetraphenylporphyrins Ana M. G. Silva Maria A. F. Faustino Tânia M. P. C. Silva Maria G. P. M. S. Neves Augusto C. Tomé Artur M. S. Silva and José A. S. Cavaleiro pg 1774; DOI: 10.1039/b203850a |
Regio- and stereocontrolled synthesis of 2-5 linked phosphorothioate oligoadenylates by uranyl ion catalyst in aqueous solution Masamitu Shimazu Kazuo Shinozuka and Hiroaki Sawai pg 1778; DOI: 10.1039/b203707f |
Regio- and stereoselective ring-opening of chiral 1,3-oxazolidin-2-one derivatives by organocopper reagents provides novel access to di-, tri- and tetra-substituted alkene dipeptide isosteres Shinya Oishi Ayumu Niida Takae Kamano Yoshihisa Miwa Tooru Taga Yoshihiko Odagaki Nobuyuki Hamanaka Mikio Yamamoto Keiichi Ajito Hirokazu Tamamura Akira Otaka and Nobutaka Fujii pg 1786; DOI: 10.1039/b203482d |
The Diels–Alder reactivity of (E)-3-phenylsulfonylprop-2-enenitrile, a cyanoacetylene equivalent Pamela J. Bradley and David H. Grayson pg 1794; DOI: 10.1039/b203391g |
Synthesis of 2,3-didehydro-2,3-dideoxy-2-fluoro apionucleosides as potential antiviral agents Hyung Ryong Moon Hea Ok Kim and Lak Shin Jeong pg 1800; DOI: 10.1039/b203126d |
Synthesis, reactivity and conformational preferences of novel enediynyl peptides: a possible scaffold for -sheet capping turns Amit Basak Kakali Rani Rudra Subhendu Sekhar Bag and Ajoy Basak pg 1805; DOI: 10.1039/b202660k |
Synthesis and lipase catalysed stereoselective acylation of some 3-methylalkan-2-ols, identified as sex pheromone precursors in females of pine sawfly species Erik Hedenström Helen Edlund Susan Lund Malin Abersten and David Persson pg 1810; DOI: 10.1039/b201395a |
Hybrid compounds generated by the introduction of a nogalamycin-producing plasmid into Streptomyces argillaceus Tero Kunnari Karel D. Klika Gloria Blanco Carmen Méndez Pekka Mäntsälä Juha Hakala Reijo Sillanpää Petri Tähtinen Jose Salas and Kristiina Ylihonko pg 1818; DOI: 10.1039/b200444p |
Irreversible photoisomerization behavior of 2-stilbazole covalently bound to porphyrin Hiroshi Sugimoto Keigo Kuramoto and Shohei Inoue pg 1826; DOI: 10.1039/b109377k |
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis Gideon Grogan Selena Guilly Ian Jackson Denise McIntyre Reuben Carr Sabine Flitsch and Nicholas Turner pg 16-vii; DOI: 10.1039/b207223h |
Chiral 2,2-bipyridines: ligands for asymmetric induction Nicholas C. Fletcher pg 1831; DOI: 10.1039/b204272j |
First synthesis of 25,26-bridged thiacalix[4]crowns by the use of a 25,26-O-disiloxanediyl-capped p-tert-butylthiacalix[4]arene Fumitaka Narumi Nobuji Matsumura Naoya Morohashi Hiroshi Kameyama and Sotaro Miyano pg 1843; DOI: 10.1039/b206050g |
A novel one pot synthesis of nitrogen containing heterocycles: an alternate methodology to the Biginelli and Hantzsch reactions Mazaahir Kidwai Shilpi Saxena Richa Mohan and R. Venkataramanan pg 1845; DOI: 10.1039/b205539m |
Some regioselective cross-coupling reactions of halopyridines and halopyrimidines Nadja M. Simkovsky Monika Ermann Stanley M. Roberts David M. Parry and Andy D. Baxter pg 1847; DOI: 10.1039/b205027g |
A concise synthesis of carpanone using solid-supported reagents and scavengers Ian R. Baxendale Ai-Lan Lee and Steven V. Ley pg 1850; DOI: 10.1039/b203388g |
Asymmetric synthesis of -pyridyl--amino acid derivatives Steven D. Bull Stephen G. Davies David. J. Fox Massimo Gianotti Peter M. Kelly Camille Pierres Edward D. Savory and Andrew D. Smith pg 1858; DOI: 10.1039/b204653a |
N-Acyl Quat pyrrolidinone auxiliary as a chiral amide equivalent via direct aminolysis Stephen G. Davies and Darren J. Dixon pg 1869; DOI: 10.1039/b205326h |
A new synthesis of temozolomide Martin J. Wanner and Gerrit-Jan Koomen pg 1877; DOI: 10.1039/b205614c |
New chiral pyrazine-based ligands for self-assembly reactions Thomas Bark Helen Stoeckli-Evans and Alexander von Zelewsky pg 1881; DOI: 10.1039/b205563p |
Efficient synthesis of N-(trifluoromethylsulfonyl)trifluoromethanesulfonimidoyl fluoride – the key agent in the preparation of compounds with superstrong electron-withdrawing groups and strong acidic properties Romute Yu. Garlyauskayte Andrey V. Bezdudny Christophe Michot Michel Armand Yurii L. Yagupolskii and Lev M. Yagupolskii pg 1887; DOI: 10.1039/b205169a |
A straightforward synthesis of DAH (3-deoxy-D-arabino-hept-2-ulosonic acid) and DRH (3-deoxy-D-ribo-hept-2-ulosonic acid) Ke-Gang Liu Shou-Gang Hu Yikang Wu Zhu-Jun Yao and Yu-Lin Wu pg 1890; DOI: 10.1039/b205047a |
Preparation and Stille cross-coupling reaction of the first organotin reagents of azulenes. Easy access to poly(azulen-6-yl)benzene derivatives Shunji Ito Tetsuo Okujima and Noboru Morita pg 1896; DOI: 10.1039/b203836f |
Synthetic transformation of hydroxymatairesinol from Norway spruce (Picea abies) to 7-hydroxysecoisolariciresinol, (+)-lariciresinol and (+)-cyclolariciresinol Patrik Eklund Reijo Sillanpää and Rainer Sjöholm pg 1906; DOI: 10.1039/b202493d |
Diastereoselective synthesis of aziridines from (1R)-10-(N,N-dialkylsulfamoyl)isobornyl 2H-azirine-3-carboxylates Yolanda S. P. Álvares M. José Alves Nuno G. Azoia Jamie F. Bickley and Thomas L. Gilchrist pg 1911; DOI: 10.1039/b202321k |
Perkin 1 Abstracts: Natural Product Synthesis Andrew Gunn Stephen McAteer Jacqueline E. Milne and Marcel de Puit pg 17-vii; DOI: 10.1039/b207912g |
Rapid analogue syntheses of heteroaromatic compounds Ian Collins pg 1921; DOI: 10.1039/b108580h |
First synthesis of phosphatidylcholine and cholesteryl derivatives bearing an unsaturated aldehyde residue Arnold N. Onyango Teruhiko Nitoda Takao Kaneko Mitsuyoshi Matsuo Shuhei Nakajima and Naomichi Baba pg 1941; DOI: 10.1039/b206231n |
Condensations of thiophene with ketones Brian J. Morrison and Oliver C. Musgrave pg 1944; DOI: 10.1039/b205484c |
Lipase-catalyzed resolution and desymmetrization of 2-hydroxymethylaziridines Paolo Davoli Emilia Caselli Maria Bucciarelli Arrigo Forni Giovanni Torre and Fabio Prati pg 1948; DOI: 10.1039/b205374h |
Synthesis of functionalised macrocyclic compounds as Na+ and K+ receptors: a mild and high yielding nitration in water of mono and bis 2-methoxyaniline functionalised crown ethers Thorfinnur Gunnlaugsson H. Q. Nimal Gunaratne Mark Nieuwenhuyzen and Joseph P. Leonard pg 1954; DOI: 10.1039/b205299g |
Synthesis and functionalization of thiophene congeners of Trger's base Tomoshige Kobayashi Takashi Moriwaki Masaya Tsubakiyama and Shihori Yoshida pg 1963; DOI: 10.1039/b205227j |
Synthesis of 2-aryl-2H,4H-imidazo[4,5-d][1,2,3]triazoles from triethyl N-(1-ethyl-2-methyl-4-nitro-1H-imidazol-5-yl)phosphorimidate by reaction with aryl isocyanates Abutariq Taher Sandra Eichenseher Alexandra M. Z. Slawin George Tennant and George W. Weaver pg 1968; DOI: 10.1039/b205216b |
Chemoenzymic synthesis of oligosaccharide fragments of the capsular polysaccharide of Streptococcus pneumoniae type 14 Dirk Michalik Johannes F. G. Vliegenthart and Johannis P. Kamerling pg 1973; DOI: 10.1039/b204933c |
Complex tetrahydrofurans from carbohydrate lactones: THF amino acids as building blocks for unnatural biopolymers Daniel D. Long Martin D. Smith Angeles Martín Joseph R. Wheatley David G. Watkin Mattaius Müller and George W. J. Fleet pg 1982; DOI: 10.1039/b111258a |
On the steric acceleration of ene reactions Nandeo Choony Nikolai Kuhnert Peter G. Sammes Graham Smith and Robert W. Ward pg 1999; DOI: 10.1039/b204778k |
Carotenoids and related polyenes. Part 9. Total synthesis of thermozeaxanthin and thermocryptoxanthin and the stabilizing effect of thermozeaxanthin on liposomes Yumiko Yamano Yoshitsugu Sakai Masayuki Hara and Masayoshi Ito pg 2006; DOI: 10.1039/b204011p |
The azomethine ylide strategy for -lactam synthesis. Azapenams and 1-azacephams David Brown Giles A. Brown Mark Andrews Jonathan M. Large Dominique Urban Craig P. Butts Neil J. Hales and Timothy Gallagher pg 2014; DOI: 10.1039/b203890k |
Synthesis and crystal structure of [26,27-2H6] 24-epi-cathasterone Adelheid Kolbe Petra Fuchs Andrea Porzel Ute Baumeister Alfred Kolbe and Günter Adam pg 2022; DOI: 10.1039/b203323b |
Book Reviews pg 2028; DOI: 10.1039/b206722f |
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis Gideon Grogan Selena Guilly Ian Jackson Denise McIntyre Reuben Carr Sabine Flitsch and Nicholas Turner pg 18-vii; DOI: 10.1039/b208231b |
Diiodosamarium based polymerisations Seema Agarwal and Andreas Greiner pg 2033; DOI: 10.1039/b203903f |
The chalcogeno-Baylis–Hillman reaction of ketones and -dicarbonyl compounds Tadashi Kataoka Hironori Kinoshita Sayaka Kinoshita and Tatsunori Iwamura pg 2043; DOI: 10.1039/b207646m |
1,2,4-Dithiazolidine-3,5-dione as an isocyanate equivalent in the Mitsunobu reaction Mark E. Wood Daniel J. Cane-Honeysett and Michael D. Dowle pg 2046; DOI: 10.1039/b206793e |
2,2,6,6-Tetramethylpiperidin-1-ylthiyl, the sulfur analogue of TEMPO, as an initiator for the controlled radical polymerisation of styrene Neil Bricklebank and Andrew Pryke pg 2048; DOI: 10.1039/b206842g |
Synthesis of Boc-protected cis- and trans-4-trifluoromethyl-D-prolines Xiao-long Qiu and Feng-ling Qing pg 2052; DOI: 10.1039/b206719f |
The development and application of ruthenium catalysed oxidations of a hydroxamic acid and in situ Diels–Alder trapping of the acyl nitroso derivative Kevin R. Flower Andrew P. Lightfoot Hayley Wan and Andrew Whiting pg 2058; DOI: 10.1039/b206430h |
A simple method for the preparation of 3-hydroxyiminodehydroquinate, a potent inhibitor of type II dehydroquinase Christine Le Sann Chris Abell and Andrew D. Abell pg 2065; DOI: 10.1039/b206066c |
Tungstate-exchanged Mg-Al-LDH catalyst: an eco-compatible route for the oxidation of sulfides in aqueous medium B. M. Choudary B. Bharathi Ch. Venkat Reddy and M. Lakshmi Kantam pg 2069; DOI: 10.1039/b205292j |
Synthesis of a pentasaccharide derivative corresponding to a triterpenoid saponin isolated from Spergularia ramosa Guofeng Gu and Yuguo Du pg 2075; DOI: 10.1039/b205106k |
Stereoselective and regioselective synthesis of azepane and azepine derivatives via piperidine ring expansion Hyun-soon Chong Bishwajit Ganguly Grant A. Broker Robin D. Rogers and Martin W. Brechbiel pg 2080; DOI: 10.1039/b204677f |
Homologation of -amino acids to -amino acids using Boc2O Ganga-Ramu Vasanthakumar Basanagoud S. Patil and Vommina V. Suresh Babu pg 2087; DOI: 10.1039/b204652k |
Elongated phosphoranes by C–C coupling of haloaroylmethylidenetriphenylphosphoranes: synthesis and applications Thies Thiemann Kuniharu Umeno Jian Wang Yumiko Tabuchi Kazuya Arima Masataka Watanabe Yasuko Tanaka Hideki Gorohmaru and Shuntaro Mataka pg 2090; DOI: 10.1039/b202745n |
Palladium-mediated synthesis of [carbonyl-11C]amides and hydrazides using [11C]carbon monoxide Farhad Karimi and Bengt Långström pg 2111; DOI: 10.1039/b202503e |
Synthesis of terminal monofluoro olefins Jan Hein van Steenis and Arne van der Gen pg 2117; DOI: 10.1039/b106187a |
Diastereoselective radical allylation and hydrogenation of -(arylsulfinyl)alkyl radicals induced by chelation control Nobuyuki Mase Yoshihiko Watanabe Koji Higuchi Shuichi Nakamura and Takeshi Toru pg 2134; DOI: 10.1039/b207249a |
Palladium-catalyzed tandem C,N-arylation of immobilized enamine for solid phase indole synthesis Kazuo Yamazaki Yosuke Nakamura and Yoshinori Kondo pg 2137; DOI: 10.1039/b206378f |
Regioselective synthesis of heterocycles by sigmatropic rearrangement: passage to 3,11a-dimethyl-6a,11a-dihydro-1H,6H-pyrano[3,4:5,6]thiopyrano[4,3-b][1]benzofuran-1-one Krishna C. Majumdar Uday K. Kundu and Subhojit Ghosh pg 2139; DOI: 10.1039/b206287a |
Diastereoselective [2,3]-sigmatropic rearrangements of lithium N-benzyl-O-allylhydroxylamides bearing a stereogenic centre adjacent to the migration terminus Steven D. Bull Stephen G. Davies Sara Hernández Domíngez Simon Jones Anne J. Price Thomas G. R. Sellers and Andrew D. Smith pg 2141; DOI: 10.1039/b207069n |
Optical resolution and racemization of areneseleninic acids Toshio Shimizu Yusuke Nakashima Itaru Watanabe Kazunori Hirabayashi and Nobumasa Kamigata pg 2151; DOI: 10.1039/b206859c |
Synthesis of (R)-6,7-dihydro-5-HETE lactone and (S)-6,7-dihydro-5-HETE lactone by using novel yeast reduction as a key reaction Satoshi Yamauchi Kenji Takeda Makoto Ganaha and Yoshiro Kinoshita pg 2156; DOI: 10.1039/b206843p |
Synthesis of nojirimycin C-glycosides Laura Cipolla Amalia Palma Barbara La Ferla and Francesco Nicotra pg 2161; DOI: 10.1039/b206623h |
Mechanistic investigations in diastereoselective Diels–Alder additions of chiral 9-anthrylethanol derivatives J. C. Christian Atherton and Simon Jones pg 2166; DOI: 10.1039/b206523a |
Synthesis of phosphorylated fragments of Streptococcus pneumoniae type 19F capsular polysaccharide Giuseppina Soliveri Anna Bertolotti Luigi Panza Laura Poletti Christopher Jones and Luigi Lay pg 2174; DOI: 10.1039/b205684d |
Synthesis and structural elucidation of 1-(3-C-ethynyl-4-thio--D-ribofuranosyl)cytosine (4-thioECyd) Noriaki Minakawa Daisuke Kaga Yuka Kato Kanji Endo Motohiro Tanaka Takuma Sasaki and Akira Matsuda pg 2182; DOI: 10.1039/b204993g |
Elemental fluorine. Part 14. Electrophilic fluorination and nitrogen functionalisation of hydrocarbons Richard D. Chambers Alan M. Kenwright Mandy Parsons Graham Sandford and John S. Moilliet pg 2190; DOI: 10.1039/b204776b |
The preparation of polymer beads by photocationic suspension co-polymerisation of 2-(arylsilyl)ethyl vinyl ethers Laurent Porres Hervé Deleuze and Yannick Landais pg 2198; DOI: 10.1039/b201520j |
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis Gideon Grogan Selena Guilly Ian Jackson Denise McIntyre Reuben Carr Sabine Flitsch and Nicholas Turner pg 20-vii; DOI: 10.1039/b209294h |
Heterogeneous and solid supported dendrimer catalysts Amy S. H. King and Lance J. Twyman pg 2209; DOI: 10.1039/b204207j |
O-Glycosylations under neutral or basic conditions Knud J. Jensen pg 2219; DOI: 10.1039/b110071h |
Expedient method for the solid-phase synthesis of some 4-substituted-4,5-dihydropyridazin-3(2H)-ones Nicolas Gouault Jean-François Cupif Maryvonne Amoros and Michèle David pg 2234; DOI: 10.1039/b205607k |
A mild, enantioselective synthesis of (R)-salmeterol via sodium borohydride–calcium chloride asymmetric reduction of a phenacyl phenylglycinol derivative Robert N. Bream Steven V. Ley Benjamin McDermott and Panayiotis A. Procopiou pg 2237; DOI: 10.1039/b207068p |
Total synthesis of (+)-curacin A, a novel antimitotic metabolite from a cyanobacterium James C. Muir Gerald Pattenden and Tao Ye pg 2243; DOI: 10.1039/b206796j |
Synthesis and antifouling activity of 3-isocyanotheonellin and its analogues Yoshikazu Kitano Toshihiro Ito Takehiro Suzuki Yasuyuki Nogata Kyouji Shinshima Erina Yoshimura Kazuhiro Chiba Masahiro Tada and Isamu Sakaguchi pg 2251; DOI: 10.1039/b206705f |
Palladium-mediated carboxylation of aryl halides (triflates) or benzyl halides using [13C]/[11C]carbon monoxide with tetrabutylammonium hydroxide or trimethylphenylammonium hydroxide Farhad Karimi and Bengt Långström pg 2256; DOI: 10.1039/b206420k |
The synthesis of benzylphosphine oxides via vicarious nucleophilic substitution and alkenes via VNS–Horner–Wittig reactions Nicholas J. Lawrence John Liddle and David Jackson pg 2260; DOI: 10.1039/b206144a |
Synthesis, structure, and reactivity of (triphenylarsoranylidene)methylcyclohepta-2,4,6-trienone derivatives: reactions with heterocumulenes and an activated acetylene Yuhki Mitsumoto and Makoto. Nitta pg 2268; DOI: 10.1039/b205612g |
Synthesis of 16-fluoro ICI 182,780 derivatives: powerful antiestrogens to image estrogen receptor densities in breast cancer by positron emission tomography Yann Seimbille François Bénard and Johan E. van Lier pg 2275; DOI: 10.1039/b205571f |
Stereochemically controlled synthesis of substituted 1,2-oxathianes Jason Eames Nikolai Kuhnert and Stuart Warren pg 2282; DOI: 10.1039/b205060a |
Hydroxy group interactions in stannylated carbohydrates. Structures and thermal stabilities of 5-deoxy-5-C-(Ph3Sn)-1,2-O-isopropylidene--D-xylofuranose, 5-deoxy-5-C-(IPh2Sn)-1,2-O-isopropylidene--D- and -L-xylofuranose, and 5-deoxy-5-C-(I2PhSn)-1,2-O-isopropylidene--D- and -L-xylofuranose Lynne A. Burnett Vitor F. Ferreira R. Alan Howie Helena Rufino Janet M. S. Skakle James L. Wardell and Solange M. S. V. Wardell pg 2288; DOI: 10.1039/b204675j |
Saturated oxygen heterocycles Mark C. Elliott pg 2301; DOI: 10.1039/b201515n |
Recent developments in the synthesis of furan-2(5H)-ones Neil B. Carter Adam E. Nadany and J.B. Sweeney pg 2324; DOI: 10.1039/b007664n |
Reaction between isocyanides and dialkyl acetylenedicarboxylates in the presence of 3-methylcyclopentane-1,2,4-trione. One-pot diastereoselective synthesis of tetrahydrocyclopenta[b]pyran derivatives Issa Yavari Mehdi Adib and Mohammad H. Sayahi pg 2343; DOI: 10.1039/b207548m |
Novel cryptands containing thiourea units as a part of the macrocyclic framework Nikolay G. Lukyanenko Tatiana I. Kirichenko and Sergey V. Scherbakov pg 2347; DOI: 10.1039/b207902j |
Nucleophilic addition reactions of bridged triene 6-chromiumtricarbonyl complexes Rohan E. J. Beckwith Michael B. Gravestock and Nigel S. Simpkins pg 2352; DOI: 10.1039/b207708f |
Reactions of 2-[(2-arylimino-2-cyano-1,1-dimethylethyl)arylamino]-3-methylbut-2-enenitrile with copper(II) acetate: synthesis of 2-(2,3-dihydro-2,2-dimethyl-3-oxo-1H-indol-1-yl)-3-methylbut-2-enenitriles Sangmin Yun and Kyongtae Kim pg 2360; DOI: 10.1039/b207530j |
A flexible synthesis of cyclopentitol derivatives based on ring-closing metathesis of carbohydrate-derived 1,6-dienes Huib Ovaa Bas Lastdrager Jeroen D. C. Codée Gijs A. van der Marel Herman S. Overkleeft and Jacques H. van Boom pg 2370; DOI: 10.1039/b207509a |
Chiral oxime ethers in asymmetric synthesis. Part 5. Asymmetric synthesis of 2-substituted 5- to 8-membered nitrogen heterocycles by oxime addition–ring-closing metathesis James C. A. Hunt Pierre Laurent and Christopher J. Moody pg 2378; DOI: 10.1039/b207235c |
Dy(OTf)3-immobilized in ionic liquids: a novel and recyclable reaction media for the synthesis of 2,3-unsaturated glycopyranosides Jhillu. S. Yadav Basi. V. Subba Reddy and J. Shyam Sunder Reddy pg 2390; DOI: 10.1039/b206957c |
Preparation of deuterium labelled fackel sterols, [5,6,6,7,7,11,11,12,12,15,16,16,17-2Hn]-5-cholesta-8,14-dien-3-ol and its (24R)-24-methyl and -ethyl congeners Hideharu Seto Keiko Mizukai Shozo Fujioka Hiroyuki Koshino and Shigeo Yoshida pg 2395; DOI: 10.1039/b206904k |
Chemo-enzymatic preparation of hydroxymethyl ketones Csaba Paizs Monica Toa Cornelia Majdik Viktória Bódai Lajos Novák Florin-Dan Irimie and László Poppe pg 2400; DOI: 10.1039/b206851f |
Sequential kinetic resolution of C2-symmetric compounds as a key step in two-directional synthesis: structural requirements for efficient resolution of difuryl diols Michael Harding Robert Hodgson and Adam Nelson pg 2403; DOI: 10.1039/b206478b |
Rhodium(II)-mediated reactions of thiobenzoylketene S,N-acetals with -diazo carbonyl compounds: synthesis of 2-substituted 3-alkylamino-5-phenylthiophenes Hyun Min Song and Kyongtae Kim pg 2414; DOI: 10.1039/b203931a |
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis Gideon Grogan Selena Guilly Ian Jackson Denise McIntyre Reuben Carr Sabine Flitsch and Nicholas Turner pg 22-ix; DOI: 10.1039/b210651p |
1,3-Dipolar cycloaddition reactions of carbohydrate derived nitrones and oximes Helen M.I. Osborn Natasha Gemmell and Laurence M. Harwood pg 2419; DOI: 10.1039/b200549m |
A chemoenzymatic synthesis of (–)-hirsutene from toluene Martin G. Banwell Alison J. Edwards Gwion J. Harfoot and Katrina A. Jolliffe pg 2439; DOI: 10.1039/b208778b |
Chiral glycine cation equivalents: N-acyliminium species derived from diketopiperazines Steven D. Bull Stephen G. Davies A. Christopher Garner Michael D. O'Shea Edward D. Savory and Emma J. Snow pg 2442; DOI: 10.1039/b207457p |
Regioselectivity in the ring-opening -scission of 2-phenyl-1,3-dioxan-2-yl radicals derived from bicyclic benzylidene acetals Yudong Cai Hai-Shan Dang and Brian P. Roberts pg 2449; DOI: 10.1039/b208200b |
Extension of the ring switch approach to glutamate antagonists to -lactam urethanes Diane Coe Martin Drysdale Oliver Philps Robert West and Douglas W. Young pg 2459; DOI: 10.1039/b207936d |
Halorosellins A and B, unique isocoumarin glucosides from the marine fungus Halorosellinia oceanica Maneekarn Chinworrungsee Prasat Kittakoop Masahiko Isaka Ratchada Chanphen Morakot Tanticharoen and Yodhathai Thebtaranonth pg 2473; DOI: 10.1039/b207887m |
Polysaccharide–polynucleotide complexes. Part 12. Enhanced affinity for various polynucleotide chains by site-specific chemical modification of schizophyllan Kazuya Koumoto Taro Kimura Masami Mizu Toyoki Kunitake Kazuo Sakurai and Seiji Shinkai pg 2477; DOI: 10.1039/b207553a |
A direct route to conjugated enediynes from dipropargylic sulfones by a modified one-flask Ramberg–Bcklund reaction Xiaoping Cao Yuying Yang and Xiaolong Wang pg 2485; DOI: 10.1039/b207296n |
Natural product-derived building blocks for combinatorial synthesis. Part 1. Fragmentation of natural products from myxobacteria Jutta Niggemann Katrin Michaelis Ronald Frank Norbert Zander and Gerhard Höfle pg 2490; DOI: 10.1039/b206953a |
Nitrilimine cycloadditions to MeOPEG-bounded alkenyl dipolarophiles Luisa Garanti Giorgio Molteni and Pietro Casati pg 2504; DOI: 10.1039/b206629g |
Conformationally locked aryl C-nucleosides: synthesis of phosphoramidite monomers and incorporation into single-stranded DNA and LNA (locked nucleic acid) B. Ravindra Babu Ashok K. Prasad Smriti Trikha Niels Thorup Virinder S. Parmar and Jesper Wengel pg 2509; DOI: 10.1039/b206626b |
Desulfurization of thioureas, benzimidazoline-2-thiones and 1,3-dihydro-1,3-diaryl-2-thioxopyrimidine-4,6(2H,5H)-diones with nickel boride at ambient temperature Jitender M. Khurana Gagan Kukreja and Geeti Bansal pg 2520; DOI: 10.1039/b206398k |
Origins of stereoselectivity in the chelation-controlled addition of alkyl radicals to -methylene--oxycarboxylic acid esters Hajime Nagano Satoko Toi Mikako Matsuda Tamano Hirasawa Satomi Hirasawa and Tomoko Yajima pg 2525; DOI: 10.1039/b205613p |
Asymmetric synthesis of C2-symmetric 5,6-bis(benzyloxy)cyclohexa-1,3-diene and a tricarbonyliron complex Akiko Watanabe Takao Kamahori Mariko Aso and Hiroshi Suemune pg 2539; DOI: 10.1039/b205526k |
Regiospecifically deuterated (–)-9-tetrahydrocannabivarins Spyros P. Nikas Ganesh A. Thakur and Alexandros Makriyannis pg 2544; DOI: 10.1039/b205459k |
Reactions of -electron rich 1,2,4-triazines with organolithium nucleophiles Joanna Szczepkowska-Sztolcman Andrzej Katrusiak Hanna Wójtowicz-Rajchel and Krzysztof Golankiewicz pg 2549; DOI: 10.1039/b205058g |
-Trifluoroacetylvinyl phenyl sulfoxide—synthesis, Diels–Alder reaction and computational study Arkady L. Krasovsky Serge A. Pissarev Valentine G. Nenajdenko and Elizabeth S. Balenkova pg 2554; DOI: 10.1039/b202583c |
The modified Julia olefination: alkene synthesis via the condensation of metallated heteroarylalkylsulfones with carbonyl compounds Paul R. Blakemore pg 2563; DOI: 10.1039/b208078h |
Nitro and related groups Joseph P. Adams pg 2586; DOI: 10.1039/b009711j |
Novel building blocks for crystal engineering: the first synthesis of oligo(imidazole)s Yasushi Morita Tsuyoshi Murata Satoru Yamada Makoto Tadokoro Akio Ichimura and Kazuhiro Nakasuji pg 2598; DOI: 10.1039/b208777d |
Tungstophosphoric acid (H3PW12O40) as a heterogeneous inorganic catalyst. Activation of hexamethyldisilazane (HMDS) by tungstophosphoric acid for efficient and selective solvent-free O-silylation reactions Habib Firouzabadi Nasser Iranpoor Kamal Amani and Farhad Nowrouzi pg 2601; DOI: 10.1039/b208202k |
Hydrosilylation of cinchonidine and 9-O-TMS-cinchonidine with triethoxysilane: application of 11-(triethoxysilyl)-10,11-dihydrocinchonidine as a chiral modifier in the enantioselective hydrogenation of 1-phenylpropane-1,2-dione Anna Lindholm Päivi Mäki-Arvela Esa Toukoniitty Tapani A. Pakkanen Janne T. Hirvi Tapio Salmi Dmitry Yu. Murzin Rainer Sjöholm and Reko Leino pg 2605; DOI: 10.1039/b205032c |
Exploiting multiple nucleophilic sites on pyrrole for the assembly of polyheterocyclic frameworks: application to a formal total synthesis of ()-aspidospermidine Martin G. Banwell and Jason A. Smith pg 2613; DOI: 10.1039/b208821e |
Solution phase synthesis of ISIS 2922 (Vitravene) by the modified H-phosphonate approach Colin B. Reese and Hongbin Yan pg 2619; DOI: 10.1039/b208802a |
Asymmetric synthesis of tetrahydrofurans by competitive [1,2]-phenylsulfanyl (PhS) migrations under thermodynamic control Lorenzo Caggiano David J. Fox David House Zoe A. Jones Fraser Kerr and Stuart Warren pg 2634; DOI: 10.1039/b208556a |
Asymmetric synthesis of tetrahydropyrans with competitive [1,2]-phenylsulfanyl (PhS) migrations Lorenzo Caggiano David J. Fox David House Zoe A. Jones Fraser Kerr and Stuart Warren pg 2646; DOI: 10.1039/b208557g |
Scope and limitation of the [1,2]-phenylsulfanyl (PhS) migration in the synthesis of tetrahydrofurans and tetrahydropyrans from common triol precursors David House Fraser Kerr and Stuart Warren pg 2652; DOI: 10.1039/b208558e |
Use of sodium triacetoxyborohydride in the synthesis of nitroxide biradicals Gerald M. Rosen Erika Schneider Sonya Shortkroff Pei Tsai and Carl S. Winalski pg 2663; DOI: 10.1039/b208263b |
PhSeOTf–Et3N Helmut Poleschner and Konrad Seppelt pg 2668; DOI: 10.1039/b207886b |
Synthesis of highly hindered oxepins and an azepine from bis-trityl carbenium ions: structural characterisation by NMR and X-ray crystallography Kieran A. Carey William Clegg Mark R. J. Elsegood Bernard T. Golding M. N. Stuart Hill and Howard Maskill pg 2673; DOI: 10.1039/b207108h |
Synthesis of [n]polynorbornanes with differing edge substitution: a new class of regioselectively addressable framework Frederick M. Pfeffer and Richard A. Russell pg 2680; DOI: 10.1039/b206057d |
2-Substituted-2,4-endo-dimethyl-8-oxabicyclo[3.2.1]octan-3-ones as catalysts for the asymmetric epoxidation of some alkenes with Oxone Solange Klein and Stanley M. Roberts pg 2686; DOI: 10.1039/b205946k |
Synthesis and characterisation of a suite of four chiral pyridyl alcohols derived from (–)-menthol Desmond Cunningham Eva T. Gallagher David H. Grayson Patrick J. McArdle Christina B. Storey and Deborah J. Wilcock pg 2692; DOI: 10.1039/b205872n |
Synthesis of N-methyl-N-(1-methylpropyl)-1-(2-chlorophenyl)isoquinoline-3-[11C]carboxamide ([11C-carbonyl]PK11195) and some analogues using [11C]carbon monoxide and 1-(2-chlorophenyl)isoquinolin-3-yl triflate Obaidur Rahman Tor Kihlberg and Bengt Långström pg 2699; DOI: 10.1039/b205838c |
Reinvestigation of base-induced skeletal conversion via a spirocyclic intermediate of dibenzodithiocinium derivatives and a computational study using the HF/6-31G* basis set Keiji Okada and Masato Tanaka pg 2704; DOI: 10.1039/b205588k |
Isolation and structure of cyclosenegalins A and B, novel cyclopeptides from the seeds of Annona senegalensis Alassane Wélé Yanjun Zhang Christelle Caux Jean-Paul Brouard Lionel Dubost Catherine Guette Jean-Louis Pousset Mamadou Badiane and Bernard Bodo pg 2712; DOI: 10.1039/b205035h |
Chemical consequences of fluorine substitution. Part 4. Diels–Alder reactions of fluorinated p-benzoquinones with Dane's diene. Synthesis of fluorinated D-homosteroids Michael Essers and Günter Haufe pg 2719; DOI: 10.1039/b208001j |
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis Gideon Grogan Selena Guilly Ian Jackson Denise McIntyre Reuben Carr Sabine Flitsch and Nicholas Turner pg 22-xv; DOI: 10.1039/b211566m |
The Sharpless asymmetric aminohydroxylation Jennifer A. Bodkin and Malcolm D. McLeod pg 2733; DOI: 10.1039/b111276g |
Synthesis of heterocycles by radical cyclisation W. Russell Bowman Anthony J. Fletcher and Graeme B. S. Potts pg 2747; DOI: 10.1039/b108582b |
Titanium reagents for the alkylidenation of carboxylic acid and carbonic acid derivatives Richard C. Hartley and Gordon J. McKiernan pg 2763; DOI: 10.1039/b009709h |
Nitroalkanes as nucleophiles in a self-catalytic Michael reaction Henryk Krawczyk Wojciech M. Wolf and Marcin liwiski pg 2794; DOI: 10.1039/b209302m |
A facile route to pyrroles, isoindoles and hetero fused analogues Christopher D. Gabbutt John D. Hepworth B. Mark Heron and Samantha L. Pugh pg 2799; DOI: 10.1039/b209255g |
Fluorination of -phenylsulfanyl esters using difluoroiodotoluene William B. Motherwell Michael F. Greaney and Derek A. Tocher pg 2809; DOI: 10.1039/b209079a |
Fluorination of sulfanyl amides using difluoroiodoarene reagents William B. Motherwell Michael F. Greaney Jeremy J. Edmunds and Jonathan W. Steed pg 2816; DOI: 10.1039/b209078c |
New ligands for asymmetric diethylzinc additions to aromatic aldehydes, demonstrating substrate-dependent nonlinear effects Philip C. Bulman Page Steven M. Allin Suzanne J. Maddocks and Mark R. J. Elsegood pg 2827; DOI: 10.1039/b208810j |
Stereocontrolled synthesis of glucosidic damascenone precursors Yumiko Yamano Yasuko Watanabe Naoharu Watanabe and Masayoshi Ito pg 2833; DOI: 10.1039/b208758h |
Palladium(0) catalysed and copper(I) promoted reactions of the secondary zinc reagent derived from L-threonine Ian Wilson and Richard F. W. Jackson pg 2845; DOI: 10.1039/b208667k |
A new tricyclic ring and a nitrogen–sulfur analogue of the tri-pentagon bowl: cycloaddition reactions of the unstablised 1,3,4-thiadiazolium-3-methanide 1,3-dipole: steric influences on the endo-effect: substituted pyrrolo[2,1-b]-1,3,4-thiadiazole systems: azolium 1,3-dipoles Richard N. Butler Georgina M. Smyth Patrick McArdle and Desmond Cunningham pg 2851; DOI: 10.1039/b208544p |
In situ IR and NMR spectroscopic investigation of the formation and structure of protonated diacetylketene tetrachloroaluminate Szilárd Csihony Andrea Bodor János Rohonczy and István T. Horváth pg 2861; DOI: 10.1039/b208387f |
Comparative study of base damage induced by gamma radiation and Fenton reaction in isolated DNA Sandrine Frelon Thierry Douki Alain Favier and Jean Cadet pg 2866; DOI: 10.1039/b207532f |
Synthesis of ,-disubstituted unnatural amino acid derivatives using the aza-[2,3]-Wittig sigmatropic rearrangement James C. Anderson and Sarah Skerratt pg 2871; DOI: 10.1039/b207295e |
Unusual hydrogen-bonding differences in stereoisomeric 6-C-alkylated cyclodextrins Tore Hardlei and Mikael Bols pg 2880; DOI: 10.1039/b207033m |
Synthesis and optimization of tri(propylene glycol) glycerolate diacrylate cross-linked polystyrene resin in polypeptide synthesis: role of the macromolecular support in solid phase peptide synthesis P. G. Sasikumar K. S. Kumar C. Arunan and V. N. Rajasekharan Pillai pg 2886; DOI: 10.1039/b206879f |
A nucleophilic addition ring closure [NARC]-based synthesis of (+) -nonactic acid Benjamin Fraser and Patrick Perlmutter pg 2896; DOI: 10.1039/b206656d |
Novel preparation of non-racemic 1-[-(1-azacycloalkyl)benzyl]-2-naphthols from Betti base and their application as chiral ligands in the asymmetric addition of diethylzinc to aryl aldehydes Jun Lu Xuenong Xu Shaozhong Wang Cunde Wang Yuefei Hu and Hongwen Hu pg 2900; DOI: 10.1039/b204534f |